SCHEMBL28148152

SCHEMBL28148152

COc1ccc(Cc2cncc3ccc(NC=O)nc23)cc1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 3/20 0.43
CYP11B1 P15538 7/20 0.42
CYP11B2 P19099 7/20 0.42
CYP19A1 P11511 1/20 0.39
CYP2C9 P11712 1/20 0.39
MPO P05164 1/20 0.36
PIM1 P11309 1/20 0.35
FTO Q9C0B1 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP2D6 P10635 1/20 0.35
ATM Q13315 1/20 0.35
SAE1 Q9UBE0 1/20 0.35
UBA2 Q9UBT2 1/20 0.35
CYP17A1 P05093 1/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28148153 0.75 PDE10A (0.44) PDE10ACYP11B1CYP11B2CYP19A1CYP2C9
SCHEMBL16229344 0.64 ALDH1A1 (0.56) ALDH1A1CYP2D6ATMSAE1UBA2
SCHEMBL28006249 0.64 CCR1 (0.44) ALDH1A1
SCHEMBL2325030 0.64 DEGS1 (0.48) PIM1ALDH1A1KDM4E
SCHEMBL27585500 0.62 CYP11B1 (0.51) PDE10ACYP11B1CYP11B2CYP19A1CYP2C9
SCHEMBL7837599 0.61 CYP11B1 (0.50) CYP11B1CYP11B2CYP19A1CYP2C9FTO
SCHEMBL28040110 0.61 ALDH1A1 (0.51) CYP11B1CYP11B2MPOALDH1A1CYP2D6
SCHEMBL1347929 0.60 ALDH1A1 (0.56) CYP2C9ALDH1A1SAE1UBA2KDM4E
SCHEMBL9558377 0.60 ERN1 (0.54) CYP2C9ALDH1A1SAE1UBA2KDM4E
SCHEMBL12869628 0.60 LTA4H (0.56) CYP11B1CYP11B2CYP2C9ALDH1A1SAE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106817900-A Novel naphthyridines and isoquinolin and its purposes as CDK8/19 inhibitor 默克专利有限公司 2017-06-09 CN disclosed