SCHEMBL28152166

SCHEMBL28152166

CC(C)(C)OC(=O)N1CCCCC1c1nc(-c2ccccc2)c(-c2ccccc2)[nH]1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 1/20 0.48
USP30 Q70CQ3 2/20 0.45
HPGDS O60760 3/20 0.43
CKS1B P61024 2/20 0.42
SKP1 P63208 2/20 0.42
SKP2 Q13309 2/20 0.42
PRMT5 O14744 1/20 0.41
HCRTR1 O43613 2/20 0.41
HCRTR2 O43614 2/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
TSHR P16473 1/20 0.41
KMT2A Q03164 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
UCHL1 P09936 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23247441 0.90 OPRD1 (0.44) OPRD1USP30HPGDSPRMT5HCRTR1
SCHEMBL18845574 0.86 OPRD1 (0.55) OPRD1USP30HPGDSHCRTR1HCRTR2
SCHEMBL8601591 0.86 MAPK14 (0.55)
SCHEMBL8602866 0.84 USP30 (0.45) USP30HCRTR1HCRTR2MEN1ALDH1A1
SCHEMBL14479516 0.80 OPRD1 (0.43) OPRD1USP30HCRTR1HCRTR2ALDH1A1
SCHEMBL11982069 0.80 OPRD1 (0.43) OPRD1USP30HCRTR1HCRTR2ALDH1A1
SCHEMBL12632942 0.80 CYP3A4 (0.46) USP30HCRTR1HCRTR2MEN1ALDH1A1
SCHEMBL23247964 0.80 RAB9A (0.47) HCRTR1HCRTR2
SCHEMBL28152181 0.80 RAB9A (0.47) HCRTR1HCRTR2
SCHEMBL18731202 0.79 UCHL1 (0.43) USP30HCRTR1HCRTR2MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106928126-B Amide derivative, preparation method and pharmaceutical application thereof 四川海思科制药有限公司 2019-12-20 CN disclosed
CN-106928126-A A kind of amide derivatives and preparation method thereof and application pharmaceutically 四川海思科制药有限公司 2017-07-07 CN disclosed