SCHEMBL28153404

SCHEMBL28153404

CNCc1ccc(-c2ccc3c(c2)CCc2c-3ccc3c2CCCC3)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 1/20 0.39
NCF1 P14598 2/20 0.35
PARP1 P09874 4/20 0.35
CYP19A1 P11511 2/20 0.35
HSD17B1 P14061 4/20 0.34
KCNH2 Q12809 2/20 0.33
HRH3 Q9Y5N1 1/20 0.33
DYRK3 O43781 1/20 0.33
TNKS O95271 1/20 0.33
PGR P06401 1/20 0.33
CDK1 P06493 1/20 0.33
ADRB1 P08588 1/20 0.33
POLA1 P09884 1/20 0.33
PIM1 P11309 1/20 0.33
SLC6A2 P23975 1/20 0.33
ADRA1A P35348 1/20 0.33
PTGS2 P35354 1/20 0.33
CDK16 Q00536 1/20 0.33
PDE4D Q08499 1/20 0.33
DYRK1A Q13627 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27454029 0.81 HSD17B1 (0.37) CYP19A1HSD17B1PARP10
SCHEMBL28118103 0.72 HSD17B1 (0.36) CYP19A1HSD17B1MPL
SCHEMBL28167174 0.69 HTR1A (0.33) PARP1KCNH2DYRK3TNKSPGR
SCHEMBL13184538 0.67 KDM4E (0.59) NOS1NCF1HRH3CHEK1ADRB2
SCHEMBL27346636 0.67 CES1 (0.47) CYP19A1DYRK1ASMN1; SMN2NPSR1
SCHEMBL19249393 0.66 ALDH1A1 (0.46) NCF1PRMT6SMN1; SMN2
SCHEMBL28845525 0.66 HAO1 (0.35) NCF1PARP1KCNH2HRH3ADRB1
Fluoride SCHEMBL28154422 0.65 DRD2 (0.33) KCNH2HRH3ADRB1SLC6A2ADRA1A
SCHEMBL17350026 0.65 ALDH1A1 (0.45) NCF1PRMT6SMN1; SMN2
SCHEMBL1254155 0.65 ALDH1A1 (0.49) NCF1PRMT6SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104876937-B Maleate, its medical composition and its use of 8 fluorine 2 { 4 [(methylamino) methyl] phenyl } 1,3,4,5 tetrahydrochysene 6H azepines * simultaneously ketone of [5,4,3 cd] indoles 6 辉瑞公司 2017-07-28 CN disclosed
CN-106794185-A High dose strength tablets of Rucaparib 克洛维斯肿瘤有限公司 2017-05-31 CN disclosed