SCHEMBL28167174

SCHEMBL28167174

CNCc1ccc(C2CCc3c(ccc4c3CCc3cc(F)ccc3-4)C2)cc1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.33
HTR7 P34969 1/20 0.33
HTR1D P28221 1/20 0.33
HTR1B P28222 1/20 0.33
NOS3 P29474 1/20 0.32
NOS2 P35228 1/20 0.32
HSD17B10 Q99714 1/20 0.32
SLC6A2 P23975 2/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
DYRK3 O43781 1/20 0.31
TNKS O95271 1/20 0.31
PGR P06401 1/20 0.31
CDK1 P06493 1/20 0.31
ADRB1 P08588 1/20 0.31
PARP1 P09874 1/20 0.31
POLA1 P09884 1/20 0.31
PIM1 P11309 1/20 0.31
ADRA1A P35348 1/20 0.31
PTGS2 P35354 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27741163 0.88
Fluoride SCHEMBL28154422 0.85 DRD2 (0.33) HTR1AHTR7SLC6A2SLC6A4SLC6A3
SCHEMBL28776118 0.75 HTR1A (0.30) HTR1AHTR7
SCHEMBL27571257 0.69 HTR1A (0.33) HTR1AHTR7
SCHEMBL28153404 0.69 NOS1 (0.39) SLC6A2DYRK3TNKSPGRCDK1
SCHEMBL27578937 0.68
SCHEMBL28210257 0.68 DAPK3 (0.41) HTR1AHTR7NOS3ADRA1ADYRK1A
SCHEMBL6156737 0.67 HTR1D (0.51) HTR1DHTR1BKCNH2
SCHEMBL28154367 0.66 DRD2 (0.32) HTR1AHTR7SLC6A2SLC6A4SLC6A3
SCHEMBL5684932 0.65 CYP2C9 (0.35) HTR1AHTR7HTR1DHTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104876937-B Maleate, its medical composition and its use of 8 fluorine 2 { 4 [(methylamino) methyl] phenyl } 1,3,4,5 tetrahydrochysene 6H azepines * simultaneously ketone of [5,4,3 cd] indoles 6 辉瑞公司 2017-07-28 CN disclosed