SCHEMBL28178459

SCHEMBL28178459

Cc1cc(F)ccc1OC(N)=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2C19 P33261 2/20 0.45
MAPT P10636 2/20 0.45
CYP2C9 P11712 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
MRGPRX4 Q96LA9 1/20 0.44
NOTUM Q6P988 1/20 0.40
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
SSTR4 P31391 1/20 0.38
MAPK14 Q16539 1/20 0.37
SLC9A1 P19634 1/20 0.37
PKM P14618 1/20 0.37
CARM1 Q86X55 1/20 0.36
PRMT6 Q96LA8 1/20 0.36
ALDH1A1 P00352 1/20 0.36
BRD4 O60885 1/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2913723 0.85 CYP2C19 (0.47) CYP1A2CYP3A4CYP2C19MAPTCYP2C9
SCHEMBL28396688 0.83 MRGPRX4 (0.49) CYP1A2CYP3A4CYP2C19MAPTCYP2C9
SCHEMBL2615140 0.83 ACHE (0.46) CYP1A2CYP3A4CYP2C19MAPTCYP2C9
SCHEMBL2615139 0.83 ACHE (0.46) CYP1A2CYP3A4CYP2C19MAPTCYP2C9
SCHEMBL29669768 0.81 L3MBTL1 (0.50) CYP1A2CYP3A4CYP2C19MAPTCYP2C9
SCHEMBL473085 0.81 L3MBTL1 (0.50) CYP1A2CYP3A4CYP2C19MAPTCYP2C9
SCHEMBL6172318 0.81 CES2 (0.45) CYP1A2CYP3A4CYP2C19MAPTNPSR1
SCHEMBL1100780 0.80 KDM4E (0.46) CYP1A2CYP3A4CYP2C19MAPTCYP2C9
SCHEMBL2191597 0.79 PDE10A (0.45) CYP1A2CYP3A4CYP2C19MAPTCYP2C9
SCHEMBL27580041 0.79 KEAP1 (0.44) CYP1A2CYP3A4CYP2C19CYP2C9L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107250126-B Long-acting dipeptidyl peptidase-IV inhibitor, application and preparation method thereof 四川科伦博泰生物医药股份有限公司 2019-10-25 CN disclosed
CN-107250126-A Long-acting dipeptidyl peptidase-IV inhibitor, application and preparation method thereof 四川科伦博泰生物医药股份有限公司 2017-10-13 CN disclosed