SCHEMBL28192513

SCHEMBL28192513

O=CCC(CF)c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABBR2 O75899 2/20 0.37
GABBR1 Q9UBS5 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP1A2 P05177 1/20 0.36
PKM P14618 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
CYP2C19 P33261 1/20 0.36
HTR2A P28223 3/20 0.34
HRH1 P35367 2/20 0.34
KDM4E B2RXH2 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
SRC P12931 1/20 0.32
MTNR1A P48039 1/20 0.32
MTNR1B P49286 1/20 0.32
KMT2A Q03164 1/20 0.31
LMNA P02545 2/20 0.31
MTOR P42345 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3140559 0.87 CYP2D6 (0.42) GABBR2GABBR1CYP2D6CYP1A2PKM
SCHEMBL1415533 0.79 TAAR1 (0.43) GABBR2GABBR1CYP2D6CYP1A2PKM
SCHEMBL19812664 0.79 GABBR2 (0.55) GABBR2GABBR1CYP2D6CYP1A2PKM
SCHEMBL27754646 0.79 CYP2C19 (0.40) GABBR2GABBR1CYP2D6CYP1A2PKM
SCHEMBL5705436 0.79 CYP2D6 (0.41) GABBR2GABBR1CYP2D6CYP1A2PKM
SCHEMBL4864892 0.79 CCR5 (0.45) GABBR2GABBR1CYP2D6CYP1A2PKM
SCHEMBL464510 0.79 CCR5 (0.45) GABBR2GABBR1CYP2D6CYP1A2PKM
SCHEMBL11537548 0.79 GABBR2 (0.37) GABBR2GABBR1CYP2D6CYP1A2PKM
SCHEMBL8906618 0.78 ALDH1A1 (0.39) TDP1SRCRAB9A
SCHEMBL8846223 0.78 MTNR1A (0.53) CYP1A2TAAR1MTNR1AMTNR1BKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107406451-A Pyrrolopyrimidines and pyrazolopyrimidines as ubiquitin-specific protease 7 inhibitors 福马治疗股份有限公司 2017-11-28 CN claimed
CN-110088096-A Piperidine derivatives as inhibitors of ubiquitin-specific protease 7 阿尔麦克探索有限公司 2019-08-02 CN disclosed
CN-107406451-A Pyrrolopyrimidines and pyrazolopyrimidines as ubiquitin-specific protease 7 inhibitors 福马治疗股份有限公司 2017-11-28 CN disclosed