SCHEMBL28200484

SCHEMBL28200484

[CH2]Cc1cc2c(Br)cccc2n1S(=O)(=O)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 1/20 0.44
HTR6 P50406 10/20 0.41
SRC P12931 1/20 0.41
CA12 O43570 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
HTR1A P08908 1/20 0.38
DRD2 P14416 1/20 0.38
HTR1D P28221 1/20 0.38
HTR1B P28222 1/20 0.38
HTR1F P30939 1/20 0.38
HTR7 P34969 1/20 0.38
DRD3 P35462 1/20 0.38
AGTR1 P30556 1/20 0.38
PSEN1 P49768 3/20 0.37
PSEN2 P49810 3/20 0.37
APH1B Q8WW43 3/20 0.37
NCSTN Q92542 3/20 0.37
APH1A Q96BI3 3/20 0.37
PSENEN Q9NZ42 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4543865 0.86 MTNR1B (0.47) MTNR1BHTR6SRCHTR1ADRD2
SCHEMBL4540819 0.81 MTNR1B (0.45) MTNR1BHTR6SRCHTR1ADRD2
SCHEMBL597369 0.80 HTR6 (0.46) HTR6SRCCA12CA2CA9
SCHEMBL30644289 0.80 HTR6 (0.46) HTR6SRCCA12CA2CA9
SCHEMBL31304851 0.79 HTR6 (0.44) HTR6SRCCA12CA2CA9
SCHEMBL16812952 0.77 HTR6 (0.48) MTNR1BHTR6SRCHTR1ADRD2
SCHEMBL25176785 0.76 RAPGEF4 (0.50) MTNR1BHTR6AGTR1PSEN1PSEN2
SCHEMBL4859176 0.76 HTR6 (0.41) MTNR1BHTR6SRCCA12CA2
SCHEMBL2431470 0.76 HTR6 (0.50) HTR6SRCAGTR1PSEN1PSEN2
SCHEMBL4852200 0.75 HTR6 (0.49) MTNR1BHTR6SRCHTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105814035-B Bruton's tyrosine kinase inhibitor 豪夫迈·罗氏有限公司 2018-02-02 CN disclosed