SCHEMBL4540819

SCHEMBL4540819

CS(=O)(=O)OCc1cc2c(Br)cccc2n1S(=O)(=O)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 1/20 0.45
HTR6 P50406 12/20 0.39
PSEN1 P49768 3/20 0.38
PSEN2 P49810 3/20 0.38
APH1B Q8WW43 3/20 0.38
NCSTN Q92542 3/20 0.38
APH1A Q96BI3 3/20 0.38
PSENEN Q9NZ42 3/20 0.38
SRC P12931 1/20 0.37
HTR1A P08908 1/20 0.37
DRD2 P14416 1/20 0.37
HTR1D P28221 1/20 0.37
HTR1B P28222 1/20 0.37
HTR1F P30939 1/20 0.37
HTR7 P34969 1/20 0.37
DRD3 P35462 1/20 0.37
AGTR1 P30556 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4543865 0.81 MTNR1B (0.47) MTNR1BHTR6PSEN1PSEN2APH1B
SCHEMBL28200484 0.81 MTNR1B (0.44) MTNR1BHTR6PSEN1PSEN2APH1B
SCHEMBL3417907 0.81 PTGDR2 (0.41) MTNR1BHTR6SRCCYP1A2CYP3A4
SCHEMBL30644289 0.78 HTR6 (0.46) HTR6PSEN1PSEN2APH1BNCSTN
SCHEMBL597369 0.78 HTR6 (0.46) HTR6PSEN1PSEN2APH1BNCSTN
SCHEMBL10004275 0.74 NOD2 (0.60) MTNR1BHTR6PSEN1PSEN2APH1B
SCHEMBL25176785 0.74 RAPGEF4 (0.50) MTNR1BHTR6PSEN1PSEN2APH1B
SCHEMBL31304851 0.74 HTR6 (0.44) HTR6SRCAGTR1
SCHEMBL4859176 0.74 HTR6 (0.41) MTNR1BHTR6SRCHTR1ADRD2
SCHEMBL4852200 0.73 HTR6 (0.49) MTNR1BHTR6PSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009112475-A1 PYRROLO [2, 3-B] PYRIDIN DERIVATIVES AS IKK2 INHIBITORS GLAXO GROUP LIMITED (GB) 2009-09-17 WO disclosed