SCHEMBL28210229

SCHEMBL28210229

O=Nc1ccc(C(=O)O)c(C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.46
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
HPGD P15428 2/20 0.43
HSD17B10 Q99714 2/20 0.43
ASPH Q12797 1/20 0.42
MEN1 O00255 1/20 0.39
PDE4A P27815 1/20 0.39
BLVRB P30043 1/20 0.39
KDR P35968 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
GRIK1 P39086 1/20 0.38
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38
USP2 O75604 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
HTR3A P46098 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28850888 0.86 CES2 (0.43) CES2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL21121922 0.80 CES2 (0.41) CES2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL7202105 0.78 MEN1 (0.50) KDM4EALDH1A1HSD17B10MEN1PDE4A
SCHEMBL25838145 0.77 ALB (0.42) CES2KDM4EALDH1A1ASPHMEN1
SCHEMBL940864 0.76 RXRB (0.54) CES2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL31000476 0.76 RXRB (0.54) CES2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL9640565 0.76 TSHR (0.48) CES2ALDH1A1HPGDHSD17B10MEN1
SCHEMBL28176917 0.76 RXRA (0.44) RXRARXRBCYP1A2
SCHEMBL11405370 0.76 MRGPRX4 (0.39) CES2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL3036944 0.75 ASPH (0.59) CES2KDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107995912-A MAYTANSINOID DERIVATIVES, CONJUGATES THEREOF, AND METHODS OF USE 里珍纳龙药品有限公司 2018-05-04 CN disclosed
CN-107922319-A Urea derivative and its purposes 东丽株式会社 2018-04-17 CN disclosed
CN-107922320-A Urea derivative and its purposes 东丽株式会社 2018-04-17 CN disclosed