SCHEMBL2829017

SCHEMBL2829017

Cc1nc2c(N3CCCC3)cccc2c(-c2ccc(S(C)(=O)=O)cc2)c1C(=O)C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.43
MAT2A P31153 1/20 0.38
NR1H2 P55055 1/20 0.38
THRB P10828 1/20 0.36
DPP4 P27487 1/20 0.35
DPP7 Q9UHL4 1/20 0.35
PLA2G7 Q13093 1/20 0.35
MGLL Q99685 1/20 0.35
ABHD6 Q9BV23 1/20 0.35
SLC6A9 P48067 1/20 0.34
KIF18A Q8NI77 1/20 0.34
PTGS1 P23219 2/20 0.34
ALOX5 P09917 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2821527 0.99 PTGS2 (0.45) PTGS2MAT2ANR1H2THRBDPP4
SCHEMBL2821151 0.90 KIF18A (0.38) PTGS2NR1H2KIF18A
SCHEMBL2822519 0.90 PTGS2 (0.34) PTGS2MAT2ANR1H2THRBDPP4
SCHEMBL2822428 0.89 GPR119 (0.36) PTGS2NR1H2PTGS1
SCHEMBL2821184 0.88 SMN1; SMN2 (0.37) DPP4
SCHEMBL2824028 0.88 FABP3 (0.43) NR1H2
SCHEMBL2825467 0.87 KDM4E (0.38)
SCHEMBL2822062 0.87 KDM4E (0.38)
SCHEMBL2825677 0.87 FABP3 (0.45) MAT2A
SCHEMBL2821880 0.87 FABP3 (0.45) MAT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809605-B1 QUINOLINES AS ALLOSTERIC ENHANCERS OF THE GABA-B RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-11 EP claimed