SCHEMBL28219978

SCHEMBL28219978

CC(c1ccc2nnccc2c1)c1ccccc1F

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 7/20 0.35
PDE1A P54750 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
PDE3B Q13370 1/20 0.35
PDE1C Q14123 1/20 0.35
PDE3A Q14432 1/20 0.35
PDE11A Q9HCR9 1/20 0.35
PDE10A Q9Y233 1/20 0.35
CYP3A4 P08684 4/20 0.34
CYP2D6 P10635 4/20 0.34
SLC6A2 P23975 4/20 0.34
SLC6A4 P31645 4/20 0.34
SLC6A3 Q01959 4/20 0.34
KCNH2 Q12809 4/20 0.34
HDAC4 P56524 3/20 0.34
ADRA2A P08913 2/20 0.32
ADRA2B P18089 2/20 0.32
ADRA2C P18825 2/20 0.32
AKR1C3 P42330 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28860238 0.82 MET (0.47) METPDE1APDE4CPDE4DPDE3B
Quinoline SCHEMBL28220135 0.80 MET (0.46) METPDE1APDE4CPDE4DPDE3B
SCHEMBL28220522 0.79 CYP1A2 (0.44) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL12702782 0.75 NPC1 (0.42) PDE10AMAT2A
SCHEMBL28219960 0.70 NCF1 (0.44)
SCHEMBL28219982 0.70 NCF1 (0.44)
SCHEMBL18713650 0.70 SCN10A (0.42) METHDAC4
SCHEMBL20675597 0.69
SCHEMBL18713526 0.68 ALDH1A1 (0.33) ADRA2AADRA2BADRA2CMAT2A
SCHEMBL10389148 0.68 ALDH1A1 (0.41) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108137547-A It can be used as the heterocyclic compound of TNF α conditioning agent 百时美施贵宝公司 2018-06-08 CN disclosed