SCHEMBL28219982

SCHEMBL28219982

C[C@@H](c1ccc2nccc(N)c2c1)c1ccccc1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 1/20 0.44
NR4A2 P43354 2/20 0.43
CCNC P24863 1/20 0.36
CDK8 P49336 1/20 0.36
PIK3CD O00329 1/20 0.36
ABL1 P00519 1/20 0.36
EGFR P00533 1/20 0.36
HCK P08631 1/20 0.36
SRC P12931 1/20 0.36
KDR P35968 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36
MTOR P42345 1/20 0.36
PIK3CG P48736 1/20 0.36
EPHB4 P54760 1/20 0.36
PRKDC P78527 1/20 0.36
SOS2 Q07890 1/20 0.34
MAP4K4 O95819 1/20 0.34
DYRK1A Q13627 1/20 0.34
TNF P01375 5/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28219960 1.00 NCF1 (0.44) NCF1NR4A2CCNCCDK8PIK3CD
SCHEMBL28860237 0.90 NCF1 (0.44) NCF1NR4A2CCNCCDK8EGFR
SCHEMBL28860238 0.77 MET (0.47) SRCKDRHSP90AA1HSP90AB1MAPT
SCHEMBL25556184 0.77 NR4A2 (0.56) NCF1NR4A2PIK3CDABL1EGFR
Quinoline SCHEMBL28220135 0.75 MET (0.46) SRCKDRHSP90AA1HSP90AB1MAPT
SCHEMBL28219978 0.70 MET (0.35)
SCHEMBL10389148 0.69 ALDH1A1 (0.41) MEN1MAPTKMT2A
SCHEMBL4155195 0.69 NR4A2 (0.54) NCF1NR4A2PIK3CDABL1EGFR
SCHEMBL28220522 0.69 CYP1A2 (0.44) LMNAMAPT
SCHEMBL16446547 0.68 NR4A2 (0.61) NCF1NR4A2CCNCCDK8SOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108137547-A It can be used as the heterocyclic compound of TNF α conditioning agent 百时美施贵宝公司 2018-06-08 CN disclosed