Quinoline

Quinoline

SCHEMBL28220135

CC(c1ccc2ncccc2c1)c1ccccc1F.c1ccc2ncccc2c1

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 15/20 0.46
ALDH1A1 P00352 3/20 0.46
PDE1A P54750 1/20 0.46
PDE4C Q08493 1/20 0.46
PDE4D Q08499 1/20 0.46
PDE3B Q13370 1/20 0.46
PDE1C Q14123 1/20 0.46
PDE3A Q14432 1/20 0.46
PDE11A Q9HCR9 1/20 0.46
PDE10A Q9Y233 1/20 0.46
AKR1C3 P42330 1/20 0.46
AKR1C2 P52895 1/20 0.46
NPC1 O15118 1/20 0.41
POLB P06746 1/20 0.41
RAB9A P51151 1/20 0.41
SRC P12931 2/20 0.40
KDR P35968 2/20 0.40
KIT P10721 1/20 0.40
FGFR2 P21802 1/20 0.40
AXL P30530 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28860238 0.97 MET (0.47) METALDH1A1PDE1APDE4CPDE4D
SCHEMBL28219978 0.80 MET (0.35) METPDE1APDE4CPDE4DPDE3B
Quinoline SCHEMBL28241576 0.79 ALDH1A1 (0.59) METALDH1A1AKR1C3AKR1C2NPC1
SCHEMBL28220522 0.78 CYP1A2 (0.44) NPC1POLBRAB9AKDM4EMAPT
SCHEMBL28219977 0.77 MET (0.41) METNPC1KDM4ETP53MAPT
SCHEMBL28219960 0.75 NCF1 (0.44) SRCKDRHSP90AA1HSP90AB1MAPT
SCHEMBL28219982 0.75 NCF1 (0.44) SRCKDRHSP90AA1HSP90AB1MAPT
SCHEMBL30606840 0.75 ALDH1A1 (0.55) METALDH1A1PDE1APDE4CPDE4D
SCHEMBL14322835 0.74 NPC1 (0.57) METALDH1A1PDE1APDE4CPDE4D
SCHEMBL112749 0.74 ALDH1A1 (0.58) METALDH1A1AKR1C3AKR1C2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108137547-A It can be used as the heterocyclic compound of TNF α conditioning agent 百时美施贵宝公司 2018-06-08 CN disclosed