SCHEMBL2822197

SCHEMBL2822197

Cc1cc(Sc2cc(C#Cc3ccc(Cl)cc3)nc(C#Cc3ccc(Cl)cc3)c2)ccc1O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 6/20 0.43
PPARG P37231 1/20 0.37
PPARD Q03181 1/20 0.37
PPARA Q07869 1/20 0.37
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
MAOA P21397 2/20 0.36
MAOB P27338 2/20 0.36
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
ALDH1A1 P00352 1/20 0.34
PLA2G1B P04054 1/20 0.34
HSP90AA1 P07900 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
HPGD P15428 1/20 0.34
ALOX15 P16050 1/20 0.34
CYP2C19 P33261 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2822191 0.86 GRM5 (0.43) GRM5PPARGPPARDPPARATP53
SCHEMBL2827433 0.85 PPARG (0.38) GRM5PPARGPPARDPPARAHSD17B10
SCHEMBL2821758 0.82 ERN1 (0.44) GRM5FFAR1
SCHEMBL11758794 0.79 TP53 (0.45) TP53MAPTMAOAMAOBMEN1
SCHEMBL2822186 0.76 PPARD (0.43) GRM5PPARGPPARDPPARAALDH1A1
SCHEMBL2822348 0.76 PPARD (0.41) GRM5PPARDMEN1KMT2AALDH1A1
SCHEMBL2069381 0.76 PPARA (0.46) PPARGPPARDPPARAFFAR1
SCHEMBL2825493 0.73 HSP90AA1 (0.34) GRM5PPARGPPARDPPARAMEN1
SCHEMBL2827431 0.72 PPARG (0.40) GRM5PPARGPPARDPPARAFFAR1
SCHEMBL51244 0.72 TP53 (0.54) TP53MAPTMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745003-B1 NOVEL COMPOUNDS, THEIR PREPARATION AND USE HIGH POINT PHARMACEUTICALS LLC (US) 2010-10-27 EP claimed