SCHEMBL2822346

SCHEMBL2822346

[O]c1ccc(Sc2cc(C#Cc3ccc(Cl)cc3)nc(C#Cc3ccc(Cl)cc3)c2)c2c1CCC2

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 1/20 0.41
GRM5 P41594 4/20 0.36
LMNA P02545 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2C9 P11712 1/20 0.30
HPGD P15428 1/20 0.30
CYP2C19 P33261 1/20 0.30
MMP13 P45452 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2822348 0.86 PPARD (0.41) PPARDGRM5CYP2C9HPGDCYP2C19
SCHEMBL2823406 0.85 PPARD (0.43) PPARD
SCHEMBL2822191 0.77 GRM5 (0.43) PPARDGRM5LMNAHPGD
SCHEMBL2822197 0.66 GRM5 (0.43) PPARDGRM5CYP2C9HPGDCYP2C19
SCHEMBL2821756 0.62 GRM5 (0.41) GRM5
SCHEMBL2822183 0.57 PPARD (0.44) PPARDGRM5HPGD
SCHEMBL719360 0.57 LMNA (0.57) GRM5LMNACYP1A2
SCHEMBL20015814 0.57 LMNA (0.57) GRM5LMNACYP1A2
Charcoal, Activated SCHEMBL31286310 0.55 KCNH2 (0.54) GRM5LMNACYP1A2
SCHEMBL12538577 0.55 GRM5 (0.59) GRM5LMNACYP1A2CYP2C9HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745003-B1 NOVEL COMPOUNDS, THEIR PREPARATION AND USE HIGH POINT PHARMACEUTICALS LLC (US) 2010-10-27 EP claimed