SCHEMBL2829123

SCHEMBL2829123

Cc1nc2c(Br)cccc2c(-c2ccc(F)cc2)c1C(=O)C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP1 P22413 3/20 0.40
DHODH Q02127 1/20 0.39
HTT P42858 3/20 0.37
KDM4E B2RXH2 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
NPSR1 Q6W5P4 2/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
PRNP P04156 1/20 0.36
PPARG P37231 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
NR2E3 Q9Y5X4 1/20 0.36
NCOR2 Q9Y618 1/20 0.36
ALDH1A1 P00352 4/20 0.36
L3MBTL1 Q9Y468 2/20 0.35
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C19 P33261 2/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2821849 0.91 GAA (0.46) ENPP1KDM4EMEN1KMT2ANPSR1
SCHEMBL2825660 0.87 NR1H2 (0.41)
SCHEMBL2823282 0.84 ENPP1 (0.39) ENPP1DHODHHTTKDM4EMEN1
SCHEMBL2825632 0.82 ESR1 (0.37) ENPP1HTTKDM4EMEN1KMT2A
SCHEMBL2821184 0.81 SMN1; SMN2 (0.37) ENPP1DHODHHTTKDM4EMEN1
SCHEMBL2825467 0.80 KDM4E (0.38) ENPP1DHODHHTTKDM4ENPSR1
SCHEMBL2822062 0.80 KDM4E (0.38) ENPP1DHODHHTTKDM4ENPSR1
SCHEMBL2824314 0.79 ENPP1 (0.35) ENPP1DHODHHTTKDM4EMEN1
SCHEMBL2824985 0.78 HPGD (0.42) MEN1KMT2ANPSR1GAAMAPT
SCHEMBL2824330 0.77 PRNP (0.61) DHODHHTTPRNPPPARGRXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809605-B1 QUINOLINES AS ALLOSTERIC ENHANCERS OF THE GABA-B RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-11 EP claimed