SCHEMBL2823571

SCHEMBL2823571

Cc1nc2ccc(Cl)c(Cl)c2c(O)c1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.33
MAPT P10636 2/20 0.33
KDM4E B2RXH2 2/20 0.33
MEN1 O00255 1/20 0.33
USP2 O75604 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
CYP3A4 P08684 1/20 0.33
MAPK1 P28482 1/20 0.33
PDE10A Q9Y233 4/20 0.33
PDE2A O00408 3/20 0.33
PKM P14618 1/20 0.33
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2822958 0.83 KDM4E (0.35) ALDH1A1MAPTKDM4EMEN1USP2
SCHEMBL1148804 0.78 MAPT (0.40) MAPTKDM4EMEN1KMT2AL3MBTL1
SCHEMBL1148916 0.75 PTGS1 (0.35) ALDH1A1MAPTKDM4EMEN1USP2
SCHEMBL1148948 0.75 RXFP1 (0.45) ALDH1A1MAPTKDM4EMEN1USP2
SCHEMBL1149264 0.74 MEN1 (0.39) ALDH1A1MAPTKDM4EMEN1KMT2A
SCHEMBL1148871 0.74 ALDH1A1 (0.41) ALDH1A1MAPTMEN1USP2KMT2A
SCHEMBL2821043 0.73 ALDH1A1 (0.36) ALDH1A1MAPTKDM4EMEN1KMT2A
SCHEMBL28427406 0.73 PARP1 (0.33) ALDH1A1MAPTKDM4EMEN1USP2
SCHEMBL2819656 0.71 ALDH1A1 (0.36) ALDH1A1MAPTKDM4EMEN1KMT2A
SCHEMBL4749202 0.71 LMNA (0.43) ALDH1A1MAPTKDM4EKMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1386914-B1 HALOGENATED QUINOLINE DERIVATIVES AND ECTOPARASITE CONTROLLERS MEIJI SEIKA KAISHA (JP) 2010-10-27 EP disclosed
CN-1310889-C Halogen-substituted quinoline derivatives and ectoparasite control agent MEIJI SEIKA KAISHA (JP) 2007-04-18 CN disclosed
US-7022855-B2 Halogen-substituted quinoline derivatives and ectoparasite control agent MEIJI SEIKA KAISHA, LTD. (JP) 2006-04-04 US disclosed
CN-1688193-A Mixed compositions for controlling parasitic insects MEIJI SEIKA KAISHA (JP) 2005-10-26 CN disclosed
EP-1559321-A1 MIXED COMPOSITIONS FOR CONTROLLING PARASITIC INSECTS MEIJI SEIKA KAISHA LTD. (JP) 2005-08-03 EP disclosed
CN-1501918-A Halogen-substituted quinoline derivatives and ectoparasite control agent �����Ƹ���ʽ���� 2004-06-02 CN disclosed
US-20040087618-A1 Halogen-substituted quinoline derivatives and ectoparasite control agent MEIJI SEIKA KAISHA, LTD. (JP) 2004-05-06 US disclosed
US-20040077602-A1 Mixture composition for controlling ectoparasites MEIJI SEIKA KAISHA, LTD. (JP) 2004-04-22 US disclosed
EP-1386914-A1 HALOGENATED QUINOLINE DERIVATIVES AND ECTOPARASITE CONTROLLERS MEIJI SEIKA KAISHA LTD. (JP) 2004-02-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040087618-A1 Halogen-substituted quinoline derivatives and ectoparasite control agent ATL3, RABL3, RAB5C ALDH1A1 2123/4885MAPT 4564/4885KDM4E 2031/4885
US-20040077602-A1 Mixture composition for controlling ectoparasites SF3A3, PEX3, HCN3 ALDH1A1 3278/4885MAPT 4378/4885KDM4E 1688/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.