SCHEMBL28237166

SCHEMBL28237166

Cc1ccc(O[C@H]2CCN(OC(=O)C(C)(C)C)C2)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.42
SCN1A P35498 1/20 0.42
SCN2A Q99250 1/20 0.42
SCN3A Q9NY46 1/20 0.42
CHRNA7 P36544 2/20 0.40
GPR119 Q8TDV5 2/20 0.40
ACACB O00763 3/20 0.39
FPR2 P25090 2/20 0.39
PROKR1 Q8TCW9 2/20 0.39
CHRM3 P20309 3/20 0.38
CHRM2 P08172 2/20 0.38
GRIN2D O15399 1/20 0.38
GRIN3B O60391 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2A Q12879 1/20 0.38
GRIN2B Q13224 1/20 0.38
GRIN2C Q14957 1/20 0.38
GRIN3A Q8TCU5 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28277464 0.94 KMT2A (0.38) EPHX2SCN1ASCN2ASCN3ACHRNA7
SCHEMBL28328550 0.92 EPHX2 (0.46) EPHX2SCN1ASCN2ASCN3ACHRNA7
SCHEMBL27911300 0.88 CHRM3 (0.49) EPHX2ACACBCHRM3CHRM2
SCHEMBL27721841 0.88 CHRM3 (0.49) EPHX2ACACBCHRM3CHRM2
SCHEMBL27874081 0.88 CHRM3 (0.49) EPHX2ACACBCHRM3CHRM2
SCHEMBL28126238 0.80 CYP2D6 (0.55) SCN1ASCN2ASCN3A
SCHEMBL27638895 0.80 EPHX2 (0.46) EPHX2GPR119ACACBFPR2PROKR1
SCHEMBL27989232 0.78 LIPG (0.47) EPHX2ACACBGRIN1GRIN2B
SCHEMBL20179924 0.77 GPR119 (0.58) GPR119
SCHEMBL28014736 0.77 FAAH (0.42) EPHX2GPR119ACACBCHRM3CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109096274-A It can be used for treating the aryl-linking compound of human tumor, neurology and amynologic disease 比奥根MA公司 2018-12-28 CN disclosed
CN-108947913-A It can be used for treating the aryl-linking compound of human tumor, neurology and amynologic disease 比奥根MA公司 2018-12-07 CN disclosed
CN-106459002-B Biaryl compounds useful in the treatment of human oncological, neurological and immunological diseases 比奥根MA公司 2018-08-21 CN disclosed