SCHEMBL28247488

SCHEMBL28247488

CN1C(=O)C(Br)Cc2ccccc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 2/20 0.45
ADRA2A P08913 1/20 0.45
ADRA2B P18089 1/20 0.45
ADRA2C P18825 1/20 0.45
SLC6A2 P23975 1/20 0.45
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45
SLC6A4 P31645 1/20 0.45
HRH1 P35367 1/20 0.45
HTR2B P41595 1/20 0.45
KCNH2 Q12809 1/20 0.45
DRD2 P14416 1/20 0.45
DRD4 P21917 1/20 0.45
ADRA1D P25100 1/20 0.45
ADRA1B P35368 1/20 0.45
AADAT Q8N5Z0 2/20 0.44
GOT1 P17174 1/20 0.44
KYAT1 Q16773 1/20 0.44
KYAT3 Q6YP21 1/20 0.44
PYGL P06737 9/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9560256 0.80 MAPT (0.56) ADRA1AADRA2AADRA2BADRA2CSLC6A2
SCHEMBL30489337 0.80 MAPT (0.56) ADRA1AADRA2AADRA2BADRA2CSLC6A2
SCHEMBL28136177 0.79 ADRA1A (0.45) ADRA1AADRA2AADRA2BADRA2CSLC6A2
SCHEMBL28136146 0.79 DRD4 (0.51) ADRA1AADRA2AADRA2BADRA2CSLC6A2
Hydrochloric Acid SCHEMBL4800198 0.77 AADAT (0.63) ADRA1AADRA2AADRA2BADRA2CSLC6A2
SCHEMBL12340980 0.77 ADRA1A (0.44) ADRA1AADRA2AADRA2BADRA2CSLC6A2
Hydrochloric Acid SCHEMBL4800182 0.77 AADAT (0.63) ADRA1AADRA2AADRA2BADRA2CSLC6A2
SCHEMBL30489285 0.76 TSHR (0.65) ADRA1AADRA2AADRA2BADRA2CSLC6A2
SCHEMBL10695532 0.76 TSHR (0.65) ADRA1AADRA2AADRA2BADRA2CSLC6A2
SCHEMBL21339127 0.76 ADRA2A (0.67) ADRA1AADRA2AADRA2BADRA2CSLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117999259-A Iron death modulators, their preparation and use 维泰瑞隆有限公司 2024-05-07 CN disclosed
CN-105102445-B Novel dihydroquinolin-2-one derivatives as aldosterone synthase (CYP11B2 or CYP11B1) inhibitors 豪夫迈·罗氏有限公司 2018-10-23 CN disclosed