SCHEMBL28249598

SCHEMBL28249598

CC(C)(C)OC(=O)c1[c]cccc1N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM6 O15303 1/20 0.38
ALDH1A1 P00352 7/20 0.36
HSD17B10 Q99714 4/20 0.36
CFTR P13569 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
SLC7A5 Q01650 1/20 0.34
ALOX15 P16050 1/20 0.33
KDM4E B2RXH2 2/20 0.33
GLA P06280 2/20 0.33
GAA P10253 2/20 0.33
MAPT P10636 2/20 0.33
HPGD P15428 2/20 0.33
HIF1A Q16665 2/20 0.33
THRB P10828 1/20 0.33
GPR119 Q8TDV5 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3060433 0.81 ADRA1A (0.36) GRM6ALDH1A1HSD17B10CA12CA1
SCHEMBL5848687 0.81 CA12 (0.36) GRM6ALDH1A1HSD17B10CA12CA1
SCHEMBL6790765 0.81 ALDH1A1 (0.52) ALDH1A1HSD17B10CFTRCA12CA1
SCHEMBL8013581 0.77 GAA (0.32) ALDH1A1HSD17B10CFTRCA12CA1
SCHEMBL28230867 0.77 GRM6 (0.38) GRM6ALDH1A1HSD17B10CFTRCA12
SCHEMBL27749672 0.77 ALDH1A1 (0.56) GRM6ALDH1A1HSD17B10CA12CA1
SCHEMBL28030866 0.73 MTNR1A (0.35) ALDH1A1HSD17B10SLC7A5KDM4EKMT2A
SCHEMBL2730411 0.73 GRM6 (0.49) GRM6ALDH1A1HSD17B10CFTRCA12
SCHEMBL3727876 0.72 MMP2 (0.41) ALDH1A1HSD17B10CFTRALOX15KDM4E
SCHEMBL8979738 0.72 CYP3A4 (0.38) ALDH1A1HSD17B10CFTRALOX15KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109071563-A Inhibitors of bruton's tyrosine kinase and methods of use thereof 詹森药业有限公司 2018-12-21 CN disclosed
CN-108884106-A POLYCYCLIC COMPOUNDS AS INHIBITORS OF BRUTON'S TYROSINE KINASE 詹森药业有限公司 2018-11-23 CN disclosed