SCHEMBL2825660

SCHEMBL2825660

Cc1nc2c(Br)cccc2c(-c2ccc(S(C)(=O)=O)cc2)c1C(=O)C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 6/20 0.41
NR1H3 Q13133 4/20 0.38
PTGS2 P35354 5/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2827841 0.87 NR1H2 (0.41) NR1H2NR1H3PTGS2
SCHEMBL2829123 0.87 ENPP1 (0.40)
SCHEMBL2821849 0.87 GAA (0.46) NR1H2NR1H3
SCHEMBL2825639 0.85 NR1H2 (0.40) NR1H2NR1H3PTGS2
SCHEMBL2829017 0.82 PTGS2 (0.43) NR1H2PTGS2
SCHEMBL2821494 0.79 PRNP (0.57) PTGS2
SCHEMBL2821151 0.79 KIF18A (0.38) NR1H2PTGS2
SCHEMBL2826443 0.78 NR1H2 (0.35) NR1H2NR1H3PTGS2
SCHEMBL2822428 0.77 GPR119 (0.36) NR1H2NR1H3PTGS2
SCHEMBL2822519 0.77 PTGS2 (0.34) NR1H2PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809605-B1 QUINOLINES AS ALLOSTERIC ENHANCERS OF THE GABA-B RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-11 EP claimed