SCHEMBL28265446

SCHEMBL28265446

COC(=O)C=Cc1cn(-c2ccccc2)nn1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.54
NPC1 O15118 2/20 0.47
RAB9A P51151 1/20 0.45
GLA P06280 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.44
POLB P06746 2/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
HTT P42858 1/20 0.44
HDAC3 O15379 4/20 0.43
HDAC4 P56524 4/20 0.43
HDAC1 Q13547 4/20 0.43
HDAC7 Q8WUI4 4/20 0.43
HDAC2 Q92769 4/20 0.43
HDAC10 Q969S8 4/20 0.43
HDAC11 Q96DB2 4/20 0.43
HDAC8 Q9BY41 4/20 0.43
HDAC6 Q9UBN7 4/20 0.43
HDAC9 Q9UKV0 4/20 0.43
HDAC5 Q9UQL6 4/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28637947 1.00 P2RX7 (0.54) P2RX7NPC1RAB9AGLAL3MBTL1
SCHEMBL28653249 0.87 CA2 (0.47) L3MBTL1POLBALDH1A1CA12CA1
SCHEMBL28632385 0.87 CA2 (0.47) L3MBTL1POLBALDH1A1CA12CA1
SCHEMBL28643460 0.86 RAB9A (0.52) P2RX7NPC1RAB9AL3MBTL1POLB
SCHEMBL28053554 0.79 HDAC1 (0.53) P2RX7NPC1RAB9APOLBALDH1A1
SCHEMBL28621729 0.79 HDAC1 (0.50) NPC1RAB9AALDH1A1HDAC3HDAC4
SCHEMBL28638771 0.79 HDAC1 (0.50) NPC1RAB9AALDH1A1HDAC3HDAC4
SCHEMBL28261748 0.79 HDAC1 (0.50) NPC1RAB9AALDH1A1HDAC3HDAC4
SCHEMBL28645125 0.78 HDAC3 (0.53) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL28625843 0.78 HDAC3 (0.53) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108997233-A A kind of synthetic method of (Z)-configuration enester triazole compounds 陕西师范大学 2018-12-14 CN disclosed