SCHEMBL28053554

SCHEMBL28053554

O=C(/C=C\c1cn(-c2ccccc2)nn1)Nc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 7/20 0.53
HDAC2 Q92769 7/20 0.53
MMP1 P03956 4/20 0.53
MMP2 P08253 4/20 0.53
MMP9 P14780 4/20 0.53
MAOB P27338 2/20 0.53
EGFR P00533 1/20 0.53
MAOA P21397 1/20 0.53
P2RX7 Q99572 1/20 0.53
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
MAPT P10636 2/20 0.50
RAB9A P51151 2/20 0.50
MIF P14174 1/20 0.48
DEGS1 O15121 1/20 0.48
HDAC3 O15379 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC11 Q96DB2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28053632 0.91 MEN1 (0.58) HDAC1HDAC2MMP1MMP2MMP9
SCHEMBL28053718 0.80 MMP1 (0.60) HDAC1HDAC2MMP1MMP2MMP9
SCHEMBL28053715 0.80 MMP1 (0.60) HDAC1HDAC2MMP1MMP2MMP9
SCHEMBL28265446 0.79 P2RX7 (0.54) HDAC1HDAC2P2RX7MEN1KMT2A
SCHEMBL28637947 0.79 P2RX7 (0.54) HDAC1HDAC2P2RX7MEN1KMT2A
SCHEMBL9840923 0.71 MMP1 (0.73) MMP1MMP2MMP9MAOBEGFR
SCHEMBL6302448 0.71 MMP1 (0.73) MMP1MMP2MMP9MAOBEGFR
SCHEMBL6302452 0.71 MMP1 (0.73) MMP1MMP2MMP9MAOBEGFR
SCHEMBL2819653 0.70 P2RX7 (1.00) MAOAP2RX7KMT2ARAB9AMIF
N-Phenylcinnamamide SCHEMBL3667414 0.70 MMP1 (1.00) MMP1MMP2MMP9MAOBEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105272928-A Alkenyl amide triazole compound and synthetic method thereof UNIV SHAANXI NORMAL 2016-01-27 CN disclosed