SCHEMBL2825542

SCHEMBL2825542

Cc1nc2c(N3CCC(O)(c4ccccc4)CC3)cccc2c(-c2ccc(S(C)(=O)=O)cc2)c1C(=O)C(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KIF18A Q8NI77 4/20 0.35
ALDH1A1 P00352 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
PTGS2 P35354 2/20 0.34
NR1H2 P55055 1/20 0.34
MCHR1 Q99705 1/20 0.34
HSD11B1 P28845 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE11A Q9HCR9 1/20 0.33
PDE10A Q9Y233 1/20 0.33
GPR6 P46095 1/20 0.33
MAT2A P31153 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2828042 0.92 MAPT (0.37) ALDH1A1MEN1KMT2AMCHR1PDE4B
SCHEMBL2828013 0.90 ALDH1A1 (0.36) ALDH1A1MCHR1
SCHEMBL2821151 0.90 KIF18A (0.38) KIF18APTGS2NR1H2
SCHEMBL2829017 0.87 PTGS2 (0.43) KIF18APTGS2NR1H2MAT2A
SCHEMBL2821527 0.86 PTGS2 (0.45) KIF18APTGS2NR1H2MAT2A
SCHEMBL2825540 0.84 ALDH1A1 (0.39) ALDH1A1MEN1KMT2APTGS2MCHR1
SCHEMBL2822519 0.83 PTGS2 (0.34) KIF18APTGS2NR1H2MAT2A
SCHEMBL2822428 0.82 GPR119 (0.36) PTGS2NR1H2GPR6
SCHEMBL2824028 0.80 FABP3 (0.43) ALDH1A1MEN1KMT2ANR1H2
SCHEMBL2826443 0.79 NR1H2 (0.35) PTGS2NR1H2GPR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809605-B1 QUINOLINES AS ALLOSTERIC ENHANCERS OF THE GABA-B RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-11 EP claimed