SCHEMBL28282946

SCHEMBL28282946

NC(=O)c1cccnc1Nc1cccc(O)c1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.73
MAPT P10636 7/20 0.67
ALDH1A1 P00352 6/20 0.67
MEN1 O00255 6/20 0.67
KMT2A Q03164 6/20 0.67
RAB9A P51151 5/20 0.67
NPC1 O15118 4/20 0.67
KCNH2 Q12809 1/20 0.67
SMN1; SMN2 Q16637 4/20 0.62
AHR P35869 1/20 0.62
MAPK1 P28482 2/20 0.55
CHEK1 O14757 1/20 0.55
PAK4 O96013 1/20 0.55
CSNK2A2 P19784 1/20 0.55
CDK2 P24941 1/20 0.55
AKT1 P31749 1/20 0.55
MAPK8 P45983 1/20 0.55
PLK1 P53350 1/20 0.55
CSNK2B P67870 1/20 0.55
CSNK2A1 P68400 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9496511 0.84 LMNA (1.00) LMNAMAPTALDH1A1MEN1KMT2A
SCHEMBL5255345 0.84 LMNA (0.71) LMNAMAPTALDH1A1MEN1KMT2A
SCHEMBL29898238 0.84 LMNA (0.71) LMNAMAPTALDH1A1MEN1KMT2A
SCHEMBL5083062 0.84 RAB9A (0.72) LMNAMAPTALDH1A1MEN1KMT2A
SCHEMBL28949487 0.84 LMNA (0.71) LMNAMAPTALDH1A1MEN1KMT2A
SCHEMBL28309786 0.84 LMNA (0.71) LMNAMAPTALDH1A1MEN1KMT2A
SCHEMBL2714471 0.83 LMNA (0.70) LMNAMAPTALDH1A1MEN1KMT2A
SCHEMBL479805 0.83 DHODH (0.76) LMNAMAPTALDH1A1MEN1KMT2A
SCHEMBL28284428 0.82 LMNA (0.68) LMNAMAPTALDH1A1MEN1KMT2A
SCHEMBL5078978 0.81 MEN1 (0.79) LMNAMAPTALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106061967-B The nicotinamide compounds replaced through heteroaryl 百时美施贵宝公司 2019-04-19 CN claimed