SCHEMBL28309786

SCHEMBL28309786

NC(=O)c1cccnc1Nc1cccc(I)c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.71
MAPT P10636 7/20 0.65
MEN1 O00255 7/20 0.65
KMT2A Q03164 7/20 0.65
RAB9A P51151 6/20 0.65
ALDH1A1 P00352 6/20 0.65
NPC1 O15118 4/20 0.65
KCNH2 Q12809 1/20 0.65
SMN1; SMN2 Q16637 5/20 0.60
AHR P35869 1/20 0.60
DHODH Q02127 4/20 0.52
HTT P42858 2/20 0.52
PKM P14618 2/20 0.51
MAPK1 P28482 1/20 0.51
GMNN O75496 1/20 0.51
TTR P02766 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51
NFKB1 P19838 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28282946 0.84 LMNA (0.73) LMNAMAPTMEN1KMT2ARAB9A
SCHEMBL5083062 0.83 RAB9A (0.72) LMNAMAPTMEN1KMT2ARAB9A
SCHEMBL29898238 0.83 LMNA (0.71) LMNAMAPTMEN1KMT2ARAB9A
SCHEMBL5255345 0.83 LMNA (0.71) LMNAMAPTMEN1KMT2ARAB9A
SCHEMBL9496511 0.83 LMNA (1.00) LMNAMAPTMEN1KMT2ARAB9A
SCHEMBL28949487 0.83 LMNA (0.71) LMNAMAPTMEN1KMT2ARAB9A
SCHEMBL2714471 0.82 LMNA (0.70) LMNAMAPTMEN1KMT2ARAB9A
SCHEMBL479805 0.82 DHODH (0.76) LMNAMAPTMEN1KMT2ARAB9A
SCHEMBL28284428 0.81 LMNA (0.68) LMNAMAPTMEN1KMT2ARAB9A
SCHEMBL29421217 0.81 RAB9A (0.73) LMNAMAPTMEN1KMT2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105814040-B The condensed 1,4- dihydro two of inhibitor as thermal excited transcryption factor 1 dislikes ene derivative 癌症研究科技有限公司 2019-07-30 CN disclosed