SCHEMBL28289709

SCHEMBL28289709

COc1ccc(C#CCC=Cc2ccccc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.54
RAB9A P51151 1/20 0.49
PPARG P37231 1/20 0.47
NFE2L2 Q16236 1/20 0.47
KMT2A Q03164 2/20 0.43
CYP1B1 Q16678 2/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
HSPD1 P10809 1/20 0.43
TNFRSF1A P19438 1/20 0.43
MAOB P27338 1/20 0.43
HSPE1 P61604 1/20 0.43
MAPK1 P28482 1/20 0.43
RELA Q04206 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
PTGER4 P35408 1/20 0.41
PTGER3 P43115 1/20 0.41
PTGER2 P43116 1/20 0.41
APP P05067 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28289707 1.00 TRPA1 (0.54) TRPA1RAB9APPARGNFE2L2KMT2A
SCHEMBL28643001 0.84 CYP1A2 (0.47) APPCYP1A2
SCHEMBL28646802 0.76 ALDH1A1 (0.49) PPARGNFE2L2KMT2AMEN1ALDH1A1
SCHEMBL8023488 0.76 TRPA1 (0.59) TRPA1PPARGNFE2L2KMT2ACYP1B1
SCHEMBL8023490 0.76 TRPA1 (0.59) TRPA1PPARGNFE2L2KMT2ACYP1B1
SCHEMBL31453513 0.76 TRPA1 (0.63) TRPA1RAB9APPARGNFE2L2KMT2A
SCHEMBL28811444 0.75 APP (0.50) RAB9AKMT2AMEN1ALDH1A1MAPT
SCHEMBL7579606 0.75 TRPA1 (0.45) TRPA1RAB9AKMT2AMEN1ALDH1A1
SCHEMBL7579599 0.75 TRPA1 (0.45) TRPA1RAB9AKMT2AMEN1ALDH1A1
SCHEMBL702843 0.74 LTA4H (0.55) RAB9AALDH1A1MAPTAPPCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109704926-B Anticancer active molecular skeleton 1, 4-eneyne compound and preparation method and application thereof 南京工业大学 2022-02-08 CN disclosed
CN-109704926-A Anticancer active molecular skeleton 1, 4-eneyne compound and preparation method and application thereof 南京工业大学 2019-05-03 CN disclosed