SCHEMBL28291609

SCHEMBL28291609

O=COCCc1cc2cc(CO)ccc2[nH]1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 2/20 0.37
MTNR1B P49286 1/20 0.37
FFAR1 O14842 12/20 0.36
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HDAC9 Q9UKV0 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34
SIRT1 Q96EB6 1/20 0.34
NHERF1 O14745 2/20 0.34
PYGL P06737 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
BACE1 P56817 1/20 0.33
PPARG P37231 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28291596 0.89 MTNR1A (0.37) MTNR1AMTNR1BHDAC3HDAC4HDAC1
SCHEMBL28038688 0.86 KDM4E (0.40) MTNR1AMTNR1BFFAR1SMN1; SMN2
SCHEMBL28072238 0.80 LOXL2 (0.54) MTNR1AMTNR1BSMN1; SMN2
SCHEMBL27613737 0.80 LOXL2 (0.54) MTNR1AMTNR1BFFAR1SIRT1PYGL
SCHEMBL27650372 0.80 CYP19A1 (0.39) MTNR1AMTNR1BFFAR1HDAC3HDAC4
SCHEMBL27648957 0.80 CYP2A6 (0.42) MTNR1AMTNR1BSIRT1SMN1; SMN2BACE1
SCHEMBL27697394 0.80 PCSK9 (0.42) MTNR1AMTNR1B
SCHEMBL28819115 0.78 MTNR1A (0.43) MTNR1AMTNR1BHDAC2SIRT1SMN1; SMN2
SCHEMBL28872616 0.78 MMP2 (0.48) MTNR1AMTNR1BSIRT1SMN1; SMN2BACE1
SCHEMBL27488329 0.78 LOXL2 (0.50) MTNR1AMTNR1BHDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109748840-A A kind of synthetic method of 2- substituted indole derivative 中国医学科学院药物研究所 2019-05-14 CN disclosed
CN-1505613-A Substituted indoles, pharmaceutical compositions containing such indoles and their use as ppar-gamma binding agents ʷ��˿�������ȳ�ķ���޹�˾ 2004-06-16 CN disclosed