SCHEMBL28291704

SCHEMBL28291704

COC(=O)C(NC(=O)CCCCCc1ccc(Br)cc1)C(C)C

nearest known ligand 0.63

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 7/20 0.58
HDAC6 Q9UBN7 6/20 0.58
SDCBP O00560 1/20 0.45
SDC2 P34741 1/20 0.45
ITGB3 P05106 1/20 0.45
ITGA2B P08514 1/20 0.45
KMT2A Q03164 2/20 0.44
ALDH1A1 P00352 1/20 0.44
MEN1 O00255 1/20 0.43
GAA P10253 1/20 0.43
ALOX5 P09917 1/20 0.43
HDAC2 Q92769 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9296228 0.83 CASP1 (0.54) HDAC1KMT2AALDH1A1MEN1ALOX5
SCHEMBL5381881 0.78 ALDH1A1 (0.54) KMT2AALDH1A1MEN1GAAHDAC2
SCHEMBL3564467 0.78 KMT2A (0.47) HDAC1HDAC6SDCBPSDC2KMT2A
SCHEMBL9977222 0.77 HDAC1 (0.44) HDAC1HDAC6SDCBPSDC2KMT2A
SCHEMBL31589186 0.77 KMT2A (0.42) HDAC1HDAC6KMT2AMEN1
SCHEMBL8621238 0.75 FAAH (0.61) KMT2AMEN1
SCHEMBL31589279 0.75 BIRC2 (0.42) HDAC1HDAC6KMT2AALDH1A1MEN1
SCHEMBL18796564 0.75 FAAH (0.61) KMT2AMEN1
SCHEMBL8018038 0.75 FAAH (0.61) KMT2AMEN1
SCHEMBL12960584 0.75 FAAH (0.61) KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109715615-A Biaryl methyl heterocycles 蒙特利尔大学 2019-05-03 CN disclosed