SCHEMBL28291790

SCHEMBL28291790

O=C(O)c1cnc(Cl)nn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT6 Q8N6T7 1/20 0.42
KDM4E B2RXH2 6/20 0.40
NAPRT Q6XQN6 3/20 0.40
HCAR2 Q8TDS4 3/20 0.40
ALDH1A1 P00352 3/20 0.39
ALOX15 P16050 3/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
P4HTM Q9NXG6 5/20 0.39
P4HA1 P13674 1/20 0.39
MIF P14174 1/20 0.39
LMNA P02545 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ASPH Q12797 2/20 0.35
KDM8 Q8N371 2/20 0.35
KMO O15229 3/20 0.35
TSHR P16473 2/20 0.34
ACMSD Q8TDX5 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
KDM6B O15054 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18366042 0.80 ALDH1A1 (0.38) SIRT6ALDH1A1L3MBTL1TDP1MAPT
SCHEMBL29185911 0.74 KDM4E (0.41) SIRT6KDM4ENAPRTHCAR2ALDH1A1
SCHEMBL20929035 0.73 KDM4E (0.40) SIRT6KDM4ENAPRTHCAR2ALDH1A1
SCHEMBL18644698 0.73 HCAR2 (0.41) SIRT6KDM4ENAPRTHCAR2ALDH1A1
SCHEMBL70035 0.72 KDM4E (0.59) SIRT6KDM4ENAPRTHCAR2ALDH1A1
SCHEMBL19875368 0.71 CYP1A2 (0.47) KDM4EALDH1A1HPGDHSD17B10LMNA
SCHEMBL287121 0.70 SIRT6 (0.72) SIRT6KDM4ENAPRTHCAR2ALDH1A1
SCHEMBL11265141 0.70 ALOX15 (0.50) SIRT6KDM4ENAPRTHCAR2ALDH1A1
SCHEMBL30159768 0.70 SIRT6 (0.72) SIRT6KDM4ENAPRTHCAR2ALDH1A1
SCHEMBL30241953 0.70 MEN1 (0.49) KDM4ENAPRTHCAR2ALDH1A1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109641875-A DIACYLGLYCEROL ACYLTRANSFERASE 2 INHIBITORS 辉瑞公司 2019-04-16 CN disclosed