SCHEMBL28292086

SCHEMBL28292086

NC(=O)c1cc2ccc(=O)[nH]c2cn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 1/20 0.49
MAPK1 P28482 3/20 0.44
CA12 O43570 2/20 0.41
CA9 Q16790 2/20 0.41
PDE3B Q13370 2/20 0.41
PDE3A Q14432 2/20 0.41
F11 P03951 1/20 0.41
NR3C1 P04150 1/20 0.38
PGR P06401 1/20 0.38
CYP3A4 P08684 1/20 0.38
CA1 P00915 1/20 0.38
CA3 P07451 1/20 0.38
CA4 P22748 1/20 0.38
CA6 P23280 1/20 0.38
CA5A P35218 1/20 0.38
CA7 P43166 1/20 0.38
CA13 Q8N1Q1 1/20 0.38
CA14 Q9ULX7 1/20 0.38
CA5B Q9Y2D0 1/20 0.38
SYK P43405 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28447307 0.80 CA12 (0.41) MAPK1CA12CA9PDE3BPDE3A
SCHEMBL28069957 0.80 GABRA1 (0.53) LCKMAPK1CA12CA9CYP3A4
SCHEMBL29721819 0.77 LCK (0.44) LCKNR3C1PGRCYP3A4SIRT6
SCHEMBL1207795 0.77 HDAC6 (0.48) LCKSYK
Hydrochloric Acid SCHEMBL3831639 0.75 HDAC6 (0.47) LCKSYK
SCHEMBL23621219 0.73 MAPK1 (0.49) MAPK1CA12CA9PDE3BPDE3A
SCHEMBL29703091 0.73 SIRT6 (0.40) LCKPDE3BPDE3ASYKSIRT6
SCHEMBL29783036 0.73 F11 (0.55) MAPK1CA12CA9PDE3BPDE3A
SCHEMBL707460 0.73 F11 (0.55) MAPK1CA12CA9PDE3BPDE3A
SCHEMBL14494403 0.73 CA12 (0.55) MAPK1CA12CA9PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109575016-A PDE9 inhibitors and uses thereof 南京药捷安康生物科技有限公司 2019-04-05 CN disclosed