SCHEMBL28447307

SCHEMBL28447307

CN(C)C(=O)c1cc2ccc(=O)[nH]c2cn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.41
CA9 Q16790 2/20 0.41
MAPK1 P28482 2/20 0.41
PDE9A O76083 2/20 0.39
PIK3CD O00329 1/20 0.39
PIK3CA P42336 1/20 0.39
PIK3CB P42338 1/20 0.39
PI4KA P42356 1/20 0.39
PIK3CG P48736 1/20 0.39
PI4KB Q9UBF8 1/20 0.39
MAPT P10636 2/20 0.39
PDE3B Q13370 3/20 0.38
PDE3A Q14432 3/20 0.38
GCK P35557 2/20 0.38
F11 P03951 1/20 0.38
DYRK1A Q13627 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
PDE5A O76074 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28292086 0.80 LCK (0.49) CA12CA9MAPK1PDE3BPDE3A
SCHEMBL28069957 0.79 GABRA1 (0.53) CA12CA9MAPK1MAPTKDM4E
Hydrochloric Acid SCHEMBL3845059 0.78 TRPM8 (0.45) PDE9APIK3CDPIK3CAPIK3CBPI4KA
SCHEMBL14494403 0.73 CA12 (0.55) CA12CA9MAPK1MAPTPDE3B
SCHEMBL4434572 0.72 CA12 (0.43) CA12CA9MAPK1PDE9AF11
SCHEMBL2017395 0.71 CYP1A2 (0.46) PIK3CDPIK3CAPIK3CBPI4KAPIK3CG
SCHEMBL23621219 0.69 MAPK1 (0.49) CA12CA9MAPK1MAPTPDE3B
SCHEMBL707460 0.69 F11 (0.55) CA12CA9MAPK1PDE3BPDE3A
SCHEMBL3732893 0.69 MAPK1 (0.49) CA12CA9MAPK1PDE3BPDE3A
SCHEMBL29783036 0.69 F11 (0.55) CA12CA9MAPK1PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111658653-B Use of phosphodiesterase inhibitors 药捷安康(南京)科技股份有限公司 2022-09-09 CN disclosed
CN-113956252-A PDE9 inhibitors and uses thereof 药捷安康(南京)科技股份有限公司 2022-01-21 CN disclosed
CN-109575016-B PDE9 inhibitors and uses thereof 药捷安康(南京)科技股份有限公司 2022-01-04 CN disclosed
CN-111658653-A Use of phosphodiesterase inhibitors 南京药捷安康生物科技有限公司 2020-09-15 CN disclosed