SCHEMBL2830183

SCHEMBL2830183

Cc1nc(OC(=O)Nc2ccn(C)n2)c(Nc2cccc(C#N)c2)s1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
CDK4 P11802 1/20 0.38
CDK2 P24941 1/20 0.38
ALDH1A1 P00352 3/20 0.38
TP53 P04637 1/20 0.38
TSHR P16473 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HSD17B10 Q99714 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
GCK P35557 1/20 0.37
ADORA2A P29274 2/20 0.37
LMNA P02545 1/20 0.37
JAK3 P52333 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2828252 0.88 CSNK2A1 (0.35) NPC1RAB9A
SCHEMBL2829284 0.85 NPC1 (0.41) NPC1RAB9ASMN1; SMN2ALDH1A1ABCG2
SCHEMBL5200154 0.84 GRM5 (0.48) NPC1RAB9ASMN1; SMN2CDK4CDK2
SCHEMBL2828971 0.83 NPC1 (0.37) NPC1RAB9ASMN1; SMN2ALDH1A1TP53
SCHEMBL2826867 0.83 CDK4 (0.45) NPC1RAB9ASMN1; SMN2CDK4CDK2
SCHEMBL2827684 0.81 GRM5 (0.48) NPC1RAB9ATSHRJAK3
SCHEMBL2831219 0.81 NPC1 (0.37) NPC1RAB9ASMN1; SMN2ALDH1A1GCK
SCHEMBL2825870 0.81 NPC1 (0.39) NPC1RAB9ASMN1; SMN2ALDH1A1PDE4B
SCHEMBL2827806 0.80 GRM5 (0.44) NPC1RAB9ASMN1; SMN2ALDH1A1LMNA
SCHEMBL2829701 0.80 GRM5 (0.48) NPC1RAB9ASMN1; SMN2CDK4CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1844044-B1 THIAZOLE-4-CARBOXAMIDE DERIVATIVES AS MGLUR5 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-07-21 EP claimed