SCHEMBL2828971

SCHEMBL2828971

COCc1cccc(Nc2sc(C)nc2OC(=O)Nc2ccn(C)n2)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.37
RAB9A P51151 3/20 0.37
KDM1A O60341 1/20 0.37
MAOB P27338 1/20 0.37
RCOR1 Q9UKL0 1/20 0.37
SMN1; SMN2 Q16637 3/20 0.36
ALDH1A1 P00352 2/20 0.36
LMNA P02545 2/20 0.36
NOTUM Q6P988 1/20 0.35
BRD4 O60885 1/20 0.35
MAPK1 P28482 1/20 0.35
KDM4E B2RXH2 1/20 0.34
HTT P42858 1/20 0.34
RAF1 P04049 1/20 0.34
KCNH2 Q12809 1/20 0.34
MEN1 O00255 1/20 0.34
TP53 P04637 1/20 0.34
KMT2A Q03164 1/20 0.34
GRM5 P41594 1/20 0.34
JAK1 P23458 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2829284 0.91 NPC1 (0.41) NPC1RAB9AKDM1ARCOR1SMN1; SMN2
SCHEMBL5200364 0.86 GRM5 (0.46) NPC1RAB9AKDM1AMAOBRCOR1
SCHEMBL2830183 0.83 NPC1 (0.40) NPC1RAB9ASMN1; SMN2ALDH1A1LMNA
SCHEMBL2827684 0.81 GRM5 (0.48) NPC1RAB9ANOTUMGRM5JAK3
SCHEMBL2831219 0.81 NPC1 (0.37) NPC1RAB9ASMN1; SMN2ALDH1A1LMNA
SCHEMBL2829461 0.80 GRM5 (0.48) NPC1RAB9AKDM1AMAOBRCOR1
SCHEMBL2824749 0.80 MET (0.42) NPC1RAB9AKDM1AMAOBRCOR1
SCHEMBL2825870 0.80 NPC1 (0.39) NPC1RAB9ASMN1; SMN2ALDH1A1LMNA
SCHEMBL2827806 0.80 GRM5 (0.44) NPC1RAB9ASMN1; SMN2ALDH1A1LMNA
SCHEMBL2826482 0.78 NPC1 (0.40) NPC1RAB9ASMN1; SMN2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1844044-B1 THIAZOLE-4-CARBOXAMIDE DERIVATIVES AS MGLUR5 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-07-21 EP claimed