SCHEMBL28293114

SCHEMBL28293114

COC(=O)c1cc2cccc([N+](=O)[O-])c2n1CN1CCS(=O)(=O)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 1/20 0.42
ALDH1A1 P00352 7/20 0.41
MAPT P10636 4/20 0.41
MAPK1 P28482 2/20 0.41
KDM4E B2RXH2 3/20 0.41
PKM P14618 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
SIRT6 Q8N6T7 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36
CYP2C19 P33261 1/20 0.36
LMNA P02545 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
F10 P00742 1/20 0.36
HRH4 Q9H3N8 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28079176 0.88 CCR2 (0.54) CCR2ALDH1A1MAPTMAPK1F10
SCHEMBL28293100 0.73 CCR2 (0.46) CCR2ALDH1A1MAPTMAPK1KDM4E
SCHEMBL1653950 0.70 CCR2 (0.46) CCR2ALDH1A1MAPTMAPK1KDM4E
SCHEMBL7953990 0.70 TSHR (0.46) CCR2ALDH1A1MAPTKDM4EL3MBTL1
SCHEMBL26660685 0.68 CCR2 (0.44) CCR2ALDH1A1MAPTKDM4EMEN1
SCHEMBL7993476 0.67 CCR2 (0.64) CCR2ALDH1A1MAPTL3MBTL1MEN1
SCHEMBL30418401 0.67 CCR2 (0.42) CCR2ALDH1A1MAPK1KDM4EL3MBTL1
SCHEMBL3560535 0.65 NOD2 (0.48) CCR2ALDH1A1MAPTMAPK1KDM4E
SCHEMBL18640132 0.65 AKR1C4 (0.54) ALDH1A1MAPTKDM4EPKML3MBTL1
SCHEMBL17865512 0.64 XDH (0.58) ALDH1A1MAPTKDM4EPKMLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105658625-B Indole amide compounds as inhibitors of cellular necrosis 株式会社LG化学 2019-05-03 CN disclosed