SCHEMBL28293217

SCHEMBL28293217

FC(F)(F)c1ccc2c(c1)CCN=C2

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.36
PNMT P11086 4/20 0.35
PARP1 P09874 1/20 0.35
PARP10 Q53GL7 1/20 0.35
TDP2 O95551 1/20 0.35
HTR2A P28223 3/20 0.33
HTR2C P28335 3/20 0.33
HTR2B P41595 3/20 0.33
EPHX2 P34913 1/20 0.33
SCN4A P35499 1/20 0.33
KIF11 P52732 1/20 0.33
POLB P06746 1/20 0.33
MAPK10 P53779 1/20 0.32
RIPK1 Q13546 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29964358 1.00 NOTUM (0.36) NOTUMPNMTPARP1PARP10TDP2
SCHEMBL28179870 0.86 PARP1 (0.38) PNMTPARP1PARP10TDP2HTR2A
SCHEMBL28061563 0.77 KIF11 (0.46) TDP2KIF11
SCHEMBL9573203 0.76 CYP19A1 (0.33) NOTUMPARP1PARP10KMT2A
SCHEMBL30074109 0.74 PNMT (0.39) NOTUMPNMTPARP1PARP10TDP2
SCHEMBL3863140 0.72 CASP1 (0.37) MEN1KMT2A
SCHEMBL29769963 0.72 CASP1 (0.37) MEN1KMT2A
SCHEMBL30025550 0.72 ADRA2A (0.34) NOTUMPARP1PARP10POLB
SCHEMBL17288395 0.72 NOTUM (0.38) NOTUMPNMTPARP1PARP10TDP2
SCHEMBL28191945 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112094229-B Synthesis method of 6- (trifluoromethyl) isoquinoline-5-alcohol 苏州康润医药有限公司 2022-11-22 CN claimed
CN-112094229-A Synthesis method of 6- (trifluoromethyl) isoquinoline-5-alcohol 苏州康润医药有限公司 2020-12-18 CN claimed
CN-112094229-B Synthesis method of 6- (trifluoromethyl) isoquinoline-5-alcohol 苏州康润医药有限公司 2022-11-22 CN disclosed
CN-112094229-A Synthesis method of 6- (trifluoromethyl) isoquinoline-5-alcohol 苏州康润医药有限公司 2020-12-18 CN disclosed
CN-105764905-B Novel octahydro-cyclobutadieno [1, 2-c; 3, 4-c' ] dipyrrole-2-yl 豪夫迈·罗氏有限公司 2019-06-07 CN disclosed
CN-109641836-A Fluorinated 2- amino -4- (substituted amino) carbanilate derivative 赛弗卢尔生命科学公司 2019-04-16 CN disclosed