Quinoline

Quinoline

SCHEMBL28294326

CC(C)(C)OC(=O)N1CC=Cc2ccccc21.c1ccc2ncccc2c1

nearest known ligand 0.40

Full drug profile on Sugi Atlas →

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 5/20 0.38
POLB P06746 2/20 0.37
ALDH1A1 P00352 1/20 0.37
GPR119 Q8TDV5 2/20 0.36
KDM1A O60341 1/20 0.36
GRM5 P41594 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
BCHE P06276 1/20 0.36
GBA1 P04062 1/20 0.35
GRM1 Q13255 1/20 0.35
BACE1 P56817 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29380399 0.86 BCHE (0.46) GPR119KDM1AGRM5BCHEGRM1
SCHEMBL5560408 0.86 BCHE (0.46) GPR119KDM1AGRM5BCHEGRM1
Quinoline SCHEMBL28157604 0.83 ALDH1A1 (0.44) POLBALDH1A1MEN1KMT2A
Indole SCHEMBL27827279 0.79 TRPA1 (0.38) KDM1AGRM5BCHEGRM1
SCHEMBL28984504 0.79 POLB (0.43) POLBGPR119KDM1AGRM5BCHE
SCHEMBL852448 0.79 POLB (0.43) POLBGPR119KDM1AGRM5GRM1
Quinoline SCHEMBL28339254 0.76 ALDH1A1 (0.50) PDE10APOLBALDH1A1MEN1KMT2A
SCHEMBL27739868 0.73 BCHE (0.48) GPR119KDM1AGRM5BCHEGRM1
Oxindole SCHEMBL28307962 0.72 AHR (0.44) KDM1AMEN1KMT2ABCHE
SCHEMBL7112196 0.72 KDM1A (0.37) GPR119KDM1AGRM5MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109761986-A Three simultaneously ring analog derivative inhibitor, preparation method and applications 上海翰森生物医药科技有限公司 2019-05-17 CN disclosed