SCHEMBL28301285

SCHEMBL28301285

CC(c1ccccc1)n1ccnc1CC1(C=O)COC1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.40
OPRD1 P41143 4/20 0.39
OPRK1 P41145 3/20 0.39
OPRM1 P35372 1/20 0.37
ALDH1A1 P00352 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
HPGD P15428 1/20 0.34
HSD17B10 Q99714 1/20 0.34
MET P08581 2/20 0.33
PIK3CD O00329 1/20 0.32
PIK3CB P42338 1/20 0.32
PIK3CG P48736 1/20 0.32
CYP2D6 P10635 1/20 0.31
FAAH O00519 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28292973 0.73 OPRD1 (0.43) BRD4OPRD1OPRK1OPRM1ALDH1A1
SCHEMBL20508884 0.72 MEN1 (0.45) BRD4OPRD1OPRK1OPRM1ALDH1A1
SCHEMBL3763386 0.72 MEN1 (0.45) BRD4OPRD1OPRK1OPRM1ALDH1A1
SCHEMBL11260988 0.71 BRD4 (0.50) BRD4OPRD1OPRK1OPRM1ALDH1A1
SCHEMBL16136368 0.68 FPR2 (0.48) BRD4OPRD1OPRK1OPRM1ALDH1A1
SCHEMBL21238449 0.67 GABRA1 (0.63) OPRD1OPRK1ALDH1A1TDP1
SCHEMBL29706729 0.66 HTR2A (0.38) ALDH1A1HPGDCYP2D6
SCHEMBL16133639 0.65 MAPT (0.46) BRD4OPRD1OPRK1OPRM1ALDH1A1
Efetozole SCHEMBL2109012 0.65 BRD4 (0.51) BRD4OPRD1OPRK1OPRM1ALDH1A1
Efetozole SCHEMBL21698044 0.65 BRD4 (0.51) BRD4OPRD1OPRK1OPRM1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109776509-A A kind of N- substituted imidazole formate ester derivative and application thereof 成都安诺晨创医药科技有限公司 2019-05-21 CN disclosed