SCHEMBL2828252

SCHEMBL2828252

Cc1nc(OC(=O)Nc2ccn(C)n2)c(Nc2cc(F)cc(C#N)c2)s1

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CSNK2A1 P68400 1/20 0.35
RAF1 P04049 1/20 0.34
PGR P06401 1/20 0.33
NPC1 O15118 3/20 0.33
RAB9A P51151 3/20 0.33
IDH1 O75874 1/20 0.33
NTRK1 P04629 1/20 0.33
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2831219 0.91 NPC1 (0.37) RAF1NPC1RAB9ANTRK1MAPK1
SCHEMBL2830183 0.88 NPC1 (0.40) NPC1RAB9A
SCHEMBL2830074 0.85 CSNK2A1 (0.38) CSNK2A1
SCHEMBL2830071 0.84 GRM5 (0.39) RAF1NPC1RAB9ANTRK1MAPK1
SCHEMBL2826367 0.81 GRM5 (0.44) CSNK2A1IDH1
SCHEMBL2828128 0.79 NPC1 (0.38) RAF1NPC1RAB9ANTRK1
SCHEMBL2827806 0.79 GRM5 (0.44) RAF1NPC1RAB9ANTRK1MAPK1
SCHEMBL2828458 0.78 ACSS2 (0.36) RAF1NPC1RAB9A
SCHEMBL2825870 0.78 NPC1 (0.39) NPC1RAB9AMAPK1
SCHEMBL2826482 0.77 NPC1 (0.40) RAF1NPC1RAB9AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1844044-B1 THIAZOLE-4-CARBOXAMIDE DERIVATIVES AS MGLUR5 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-07-21 EP claimed