SCHEMBL28302135

SCHEMBL28302135

CC(C)(C)OC(=O)NOCCc1cccc(S(=O)(=O)NC2CC2)c1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.47
ALDH1A1 P00352 2/20 0.47
KMT2A Q03164 1/20 0.42
CA2 P00918 1/20 0.42
ACACB O00763 1/20 0.40
ALOX5 P09917 1/20 0.39
NR1H2 P55055 6/20 0.39
ADRB2 P07550 2/20 0.38
ADRB1 P08588 2/20 0.38
ADRB3 P13945 2/20 0.38
BRD4 O60885 1/20 0.38
BRD2 P25440 1/20 0.38
BRD3 Q15059 1/20 0.38
HTR1A P08908 2/20 0.38
HTR7 P34969 2/20 0.38
STS P08842 1/20 0.38
NR1H3 Q13133 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28302149 0.85 CA2 (0.43) KMT2ACA2ACACBALOX5ADRB2
SCHEMBL28302128 0.82 CA2 (0.48) LMNACA2ALOX5NR1H2
SCHEMBL3386695 0.80 LMNA (0.48) LMNAALDH1A1KMT2ACA2ACACB
SCHEMBL13400331 0.73 LMNA (0.48) LMNAALDH1A1KMT2AACACBADRB2
SCHEMBL28302172 0.73 CACNA1B (0.35) LMNAALDH1A1KMT2ACA2ACACB
SCHEMBL27885422 0.72 ALDH1A1 (0.52) LMNAALDH1A1KMT2ABRD4BRD2
SCHEMBL13469348 0.71 ALDH1A1 (0.58) LMNAALDH1A1KMT2ABRD4BRD2
SCHEMBL14249971 0.71 ALDH1A1 (0.58) LMNAALDH1A1KMT2ABRD4BRD2
SCHEMBL15899804 0.71 ALDH1A1 (0.55) LMNAALDH1A1KMT2ABRD4BRD2
SCHEMBL18151417 0.71 ALDH1A1 (0.58) LMNAALDH1A1KMT2ABRD4BRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109952298-A Indole carboxamides analog derivative, preparation method and its application in medicine 江苏恒瑞医药股份有限公司 2019-06-28 CN disclosed