SCHEMBL28320591

SCHEMBL28320591

FC(F)(F)Oc1cccc(-c2nc(-c3c[nH]nn3)cs2)c1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.43
PIM1 P11309 2/20 0.41
PIM3 Q86V86 1/20 0.41
SCN9A Q15858 3/20 0.41
EIF4E P06730 2/20 0.40
HSD17B1 P14061 1/20 0.40
HSD17B2 P37059 1/20 0.40
KCNH2 Q12809 1/20 0.40
SCN10A Q9Y5Y9 1/20 0.40
CYP19A1 P11511 1/20 0.39
LDHA P00338 1/20 0.39
SREBF2 Q12772 1/20 0.39
GRM5 P41594 1/20 0.38
DYRK1A Q13627 2/20 0.38
CYP2C9 P11712 1/20 0.38
GAA P10253 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28320520 0.85 PIM1 (0.45) PIM1EIF4ESCN10ACYP19A1
SCHEMBL28321645 0.83 ALDH1A1 (0.53) XDHPIM1EIF4EHSD17B1HSD17B2
SCHEMBL23457617 0.82 XDH (0.52) XDHPIM1PIM3KCNH2SCN10A
SCHEMBL29699351 0.82 XDH (0.52) XDHPIM1PIM3KCNH2SCN10A
SCHEMBL28321648 0.80 IDO1 (0.43) XDHPIM1SCN9AEIF4EHSD17B1
SCHEMBL28251098 0.80 KDM4E (0.52) XDHSCN9AEIF4EHSD17B1HSD17B2
SCHEMBL28321644 0.79 KCNH2 (0.43) XDHPIM1SCN9AEIF4EHSD17B1
SCHEMBL28320570 0.78 ALOX5 (0.47) PIM1EIF4ESCN10ACYP19A1GAA
SCHEMBL16399094 0.77 CTSS (0.44) XDHPIM1SCN9AEIF4ESREBF2
SCHEMBL16400544 0.77 ADORA1 (0.42) XDHPIM1SCN9AEIF4EKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105408325-B cyanotriazole compounds 大塚制药株式会社 2019-10-22 CN claimed
CN-105408325-B cyanotriazole compounds 大塚制药株式会社 2019-10-22 CN disclosed