SCHEMBL28340415

SCHEMBL28340415

O=C(O)C=CC(=O)c1ccccc1-c1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 1/20 0.59
BCAT2 O15382 1/20 0.55
MEN1 O00255 4/20 0.53
KMT2A Q03164 4/20 0.53
ALDH1A1 P00352 3/20 0.53
CYP2C9 P11712 1/20 0.53
HPGD P15428 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.50
CHRNB2 P17787 2/20 0.49
CHRNB4 P30926 2/20 0.49
CHRNA3 P32297 2/20 0.49
CHRNA4 P43681 2/20 0.49
HNF4A P41235 1/20 0.47
TSHR P16473 1/20 0.46
RECQL P46063 1/20 0.46
HSP90AA1 P07900 2/20 0.44
KDM4E B2RXH2 2/20 0.44
MAPT P10636 2/20 0.44
PKM P14618 1/20 0.44
MITF O75030 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18813656 0.85 GPR52 (0.59) GPR52BCAT2MEN1KMT2AALDH1A1
SCHEMBL27574463 0.81 MAPT (0.64) GPR52BCAT2MEN1KMT2AALDH1A1
SCHEMBL7864455 0.80 BCAT2 (0.59) GPR52BCAT2MEN1KMT2AALDH1A1
SCHEMBL28993895 0.79 RECQL (0.59) GPR52BCAT2MEN1KMT2AALDH1A1
SCHEMBL5180034 0.78 BCAT2 (0.57) GPR52BCAT2MEN1KMT2AALDH1A1
SCHEMBL31521259 0.78 BCAT2 (0.57) GPR52BCAT2MEN1KMT2AALDH1A1
Biphenyl SCHEMBL28611778 0.76 ALDH1A1 (0.63) MEN1KMT2AALDH1A1CYP2C9HPGD
Biphenyl SCHEMBL10898338 0.76 ALDH1A1 (0.63) MEN1KMT2AALDH1A1CYP2C9HPGD
Biphenyl SCHEMBL5421614 0.76 ALDH1A1 (0.63) MEN1KMT2AALDH1A1CYP2C9HPGD
Biphenyl SCHEMBL9816554 0.76 ALDH1A1 (0.63) MEN1KMT2AALDH1A1CYP2C9HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106860441-B Application of 4-oxo-2-butenamide derivative in preparation of bacteriostatic agent 中国医学科学院医药生物技术研究所 2019-12-31 CN disclosed