SCHEMBL28350517

SCHEMBL28350517

COc1cc2ncnc(Nc3cccnc3)c2cc1OCCCN1CCOCC1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 10/20 0.77
KDR P35968 8/20 0.77
EGFR P00533 6/20 0.72
BRAF P15056 2/20 0.69
LCK P06239 2/20 0.69
RET P07949 2/20 0.69
MET P08581 2/20 0.69
MAPT P10636 2/20 0.69
LTK P29376 2/20 0.69
TNK2 Q07912 2/20 0.69
MAP4K5 Q9Y4K4 2/20 0.69
EPHB4 P54760 2/20 0.69
CIT O14578 1/20 0.69
GAK O14976 1/20 0.69
EPHB6 O15197 1/20 0.69
ABCC4 O15439 1/20 0.69
DAPK3 O43293 1/20 0.69
RIPK2 O43353 1/20 0.69
NR1I2 O75469 1/20 0.69
RPS6KA4 O75676 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28354308 1.00 SRC (0.77) SRCKDREGFRBRAFLCK
SCHEMBL13529060 0.90 SRC (0.84) SRCKDREGFRBRAFLCK
SCHEMBL6165865 0.86 HDAC1 (0.73) SRCKDREGFRBRAFLCK
SCHEMBL6163849 0.86 HDAC1 (0.73) SRCKDREGFRBRAFLCK
SCHEMBL6906285 0.86 KDR (0.82) SRCKDREGFRBRAFLCK
SCHEMBL3531151 0.86 SRC (0.86) SRCKDREGFRBRAFLCK
SCHEMBL28350751 0.86 SRC (0.77) SRCKDREGFRAURKA
SCHEMBL1155807 0.85 SRC (0.81) SRCKDREGFRBRAFLCK
SCHEMBL28350757 0.85 SRC (0.73) SRCKDREGFRBRAFLCK
SCHEMBL28354714 0.85 SRC (0.73) SRCKDREGFRBRAFLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110746398-A 4-heterocyclic substituted quinazoline derivative and preparation method and application thereof 刘沛友 2020-02-04 CN disclosed