SCHEMBL2835846

SCHEMBL2835846

CN1Cc2sccc2C(O)C1

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.55
RAB9A P51151 1/20 0.55
SLC6A4 P31645 15/20 0.40
SLC6A3 Q01959 15/20 0.40
SLC6A2 P23975 14/20 0.40
CYP2D6 P10635 2/20 0.37
HHAT Q5VTY9 1/20 0.34
DRD2 P14416 1/20 0.33
DRD1 P21728 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2836823 0.82 DRD1 (0.41) NPC1RAB9AHHATDRD2DRD1
SCHEMBL2839500 0.82 NPC1 (0.46) NPC1RAB9AHHATDRD2DRD1
SCHEMBL2836800 0.77 NPC1 (0.38) NPC1RAB9ASLC6A4SLC6A3SLC6A2
SCHEMBL14970374 0.76 HHAT (0.43) NPC1RAB9AHHAT
SCHEMBL4751909 0.75 NPC1 (0.49) NPC1RAB9ASLC6A4SLC6A3SLC6A2
SCHEMBL11640087 0.74 NPC1 (0.62) NPC1RAB9ASLC6A4SLC6A3SLC6A2
SCHEMBL4751291 0.74 HHAT (0.38) NPC1RAB9AHHAT
SCHEMBL16219044 0.74 CHRNB2 (0.37) NPC1RAB9ASLC6A4HHAT
SCHEMBL15490061 0.73 OPRM1 (0.38) NPC1RAB9A
SCHEMBL2837960 0.73 SLC6A4 (0.41) NPC1RAB9ASLC6A4SLC6A3SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8217031-B2 Heteroaryl derivatives NIPPON SHINYAKU CO., LTD. (JP) 2012-07-10 US disclosed
US-20100048537-A1 HETEROARYL DERIVATIVES NIPPON SHINYAKU CO., LTD. (JP) 2010-02-25 US disclosed
EP-2141168-A1 HETEROARYL DERIVATIVES Nippon Shinyaku Co., Ltd. (JP) 2010-01-06 EP disclosed
US-4076819-A ANTIINFLAMMATORY AGENTS, INHIBITOR OF BLOOD PLATELET AGGREGATION PARCOR (FR) 1978-02-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100048537-A1 HETEROARYL DERIVATIVES OPRD1, OPRM1, OPRK1 NPC1 1665/4885RAB9A 1933/4885SLC6A4 185/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.