SCHEMBL28360893

SCHEMBL28360893

Fc1ccc[c]c1-c1cc(Cl)cc(Cl)c1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
HPGD P15428 1/20 0.35
CYP2C19 P33261 1/20 0.35
TSHR P16473 1/20 0.31
GAA P10253 1/20 0.30
AKR1C3 P42330 1/20 0.30
AKR1C2 P52895 1/20 0.30
APP P05067 1/20 0.30
NPC1 O15118 1/20 0.30
CASP3 P42574 1/20 0.30
RAB9A P51151 1/20 0.30
SENP8 Q96LD8 1/20 0.30
SENP7 Q9BQF6 1/20 0.30
SENP6 Q9GZR1 1/20 0.30
RXRA P19793 1/20 0.30
RXRB P28702 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29248267 0.88 ADORA2A (0.35)
SCHEMBL16058080 0.85 ALOX5 (0.42) TSHRNPC1RAB9A
SCHEMBL435279 0.82 CYP1A2 (0.38) L3MBTL1CYP1A2CYP2C9CYP2C19TSHR
SCHEMBL10936903 0.77 ESR2 (0.33) CYP1A2TSHRGAARXRARXRB
SCHEMBL9649078 0.77 TSHR (0.31) TSHRRXRARXRB
SCHEMBL3607306 0.75 ALDH1A1 (0.35) L3MBTL1ALDH1A1NPC1RAB9A
SCHEMBL28357115 0.75 ADORA2A (0.46)
SCHEMBL433087 0.74 EGLN2 (0.37) CYP2C9
SCHEMBL17514939 0.74 CYP1A1 (0.46) L3MBTL1ALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL28357088 0.74 ADORA2A (0.34) NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110809577-A Modulators of adenosine A2A receptor 雷沃医疗有限公司 2020-02-18 CN claimed
CN-110809577-A Modulators of adenosine A2A receptor 雷沃医疗有限公司 2020-02-18 CN disclosed