SCHEMBL28362248

SCHEMBL28362248

C=CCCC(=O)NC(CCCc1ccccc1)C(=O)OCC#N

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 4/20 0.40
CTSG P08311 1/20 0.40
CMA1 P23946 1/20 0.40
FAAH O00519 4/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
MGLL Q99685 1/20 0.39
CTSL P07711 1/20 0.39
CTSS P25774 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21895862 1.00 CASP1 (0.40) CASP1CTSGCMA1FAAHSMN1; SMN2
SCHEMBL21895861 0.94 CTSS (0.43) CASP1CTSGCMA1FAAHSMN1; SMN2
SCHEMBL21895863 0.94 CTSS (0.43) CASP1CTSGCMA1FAAHSMN1; SMN2
SCHEMBL7074221 0.87 ACE (0.47) CTSLCTSS
SCHEMBL7074223 0.87 ACE (0.47) CTSLCTSS
SCHEMBL15083124 0.86 CYP1A2 (0.36) CASP1FAAHCTSLCTSS
SCHEMBL16287223 0.86 CASP1 (0.41) CASP1CTSGCMA1FAAHSMN1; SMN2
SCHEMBL16287221 0.86 CASP1 (0.41) CASP1CTSGCMA1FAAHSMN1; SMN2
SCHEMBL16289502 0.86 CYP1A2 (0.36) CASP1FAAHCTSLCTSS
SCHEMBL16289204 0.83 CASP1 (0.33) CASP1CTSLCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118256591-A Cyclic peptide compound having high membrane permeability and library comprising same 中外制药株式会社 2024-06-28 CN disclosed
CN-110869544-B Cyclic peptide compound having high membrane permeability and library comprising same 中外制药株式会社 2024-03-08 CN disclosed
CN-110869544-A Cyclic peptide compound having high membrane permeability and library containing same 中外制药株式会社 2020-03-06 CN disclosed