SCHEMBL21895863

SCHEMBL21895863

C=CCCC(=O)NC(CCc1ccccc1)C(=O)OCC#N

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSS P25774 2/20 0.43
CTSK P43235 1/20 0.43
CASP1 P29466 4/20 0.40
CTSL P07711 3/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CNR2 P34972 1/20 0.38
CTSB P07858 1/20 0.37
CTSG P08311 2/20 0.37
CMA1 P23946 2/20 0.37
PRSS1 P07477 1/20 0.37
CTRB1 P17538 1/20 0.37
RAB9A P51151 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
FAAH O00519 2/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNA4 P43681 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21895861 1.00 CTSS (0.43) CTSSCTSKCASP1CTSLSMN1; SMN2
SCHEMBL28362248 0.94 CASP1 (0.40) CTSSCASP1CTSLSMN1; SMN2CTSG
SCHEMBL21895862 0.94 CASP1 (0.40) CTSSCASP1CTSLSMN1; SMN2CTSG
SCHEMBL21950780 0.89 CNR2 (0.36) CTSSCTSKCNR2
SCHEMBL28362291 0.89 CNR2 (0.36) CTSSCTSKCNR2
SCHEMBL7074223 0.89 ACE (0.47) CTSSCTSKCTSLCTSB
SCHEMBL7074221 0.89 ACE (0.47) CTSSCTSKCTSLCTSB
SCHEMBL21895954 0.89 CTSL (0.39) CTSSCTSKCTSLSMN1; SMN2CTSB
SCHEMBL28366266 0.89 CTSL (0.39) CTSSCTSKCTSLSMN1; SMN2CTSB
SCHEMBL21896476 0.87 CTSG (0.35) CTSSCTSKSMN1; SMN2CTSGCMA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118256591-A Cyclic peptide compound having high membrane permeability and library comprising same 中外制药株式会社 2024-06-28 CN disclosed
CN-110869544-B Cyclic peptide compound having high membrane permeability and library comprising same 中外制药株式会社 2024-03-08 CN disclosed
EP-3636807-A1 CYCLIC PEPTIDE COMPOUND HAVING HIGH MEMBRANE PERMEABILITY, AND LIBRARY CONTAINING SAME Chugai Seiyaku Kabushiki Kaisha (JP) 2020-04-15 EP disclosed
CN-110869544-A Cyclic peptide compound having high membrane permeability and library containing same 中外制药株式会社 2020-03-06 CN disclosed