SCHEMBL28390751

SCHEMBL28390751

N#CC(c1ccc(C(F)(F)F)cc1)C1CCN(C(=O)O)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 4/20 0.45
DPP7 Q9UHL4 3/20 0.45
DPP8 Q6V1X1 2/20 0.43
TEAD1 P28347 2/20 0.42
HSD11B1 P28845 1/20 0.41
GAA P10253 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
MGLL Q99685 1/20 0.40
CACNA1A O00555 1/20 0.39
CACNA2D1 P54289 1/20 0.39
CACNA1B Q00975 1/20 0.39
CACNB1 Q02641 1/20 0.39
CACNA1C Q13936 1/20 0.39
NOTUM Q6P988 1/20 0.39
FAP Q12884 1/20 0.38
DPP9 Q86TI2 1/20 0.38
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
SLC6A4 P31645 1/20 0.38
EPHX2 P34913 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28475071 0.85 CACNA1B (0.43) DPP4DPP7DPP8HSD11B1MGLL
SCHEMBL27144128 0.85 CACNA1B (0.43) DPP4DPP7DPP8HSD11B1MGLL
SCHEMBL4236045 0.83 MMP13 (0.51) DPP4
SCHEMBL15536288 0.83 FPR2 (0.49) DPP4DPP7MGLLCACNA2D1CACNA1B
SCHEMBL23212032 0.80 TEAD1 (0.50) DPP4DPP7DPP8TEAD1GAA
SCHEMBL28162309 0.80 RPS6KB1 (0.53) DPP4DPP7DPP8TEAD1GAA
SCHEMBL14638795 0.72 HSD11B1 (0.71) HSD11B1GAATDP1MGLLNOTUM
SCHEMBL21381906 0.72 GAA (0.48) DPP4DPP7TEAD1HSD11B1GAA
SCHEMBL2636716 0.72 LIPE (0.52) HSD11B1GAATDP1NOTUM
SCHEMBL17942511 0.72 ADAMTS7 (0.45) HSD11B1GAATDP1CACNA1BNOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106946796-B Aminopyrimidine derivatives useful as modulators of kinase activity 默克专利有限公司 2020-05-08 CN disclosed