SCHEMBL28408689

SCHEMBL28408689

O=C(c1ccccc1)N1CCCCC1c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.54
PARP14 Q460N5 1/20 0.50
PARP10 Q53GL7 1/20 0.50
KMT2A Q03164 3/20 0.48
HTT P42858 2/20 0.48
MAPT P10636 5/20 0.47
POLB P06746 4/20 0.47
LMNA P02545 4/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MEN1 O00255 1/20 0.47
HPGD P15428 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
CES2 O00748 1/20 0.46
CES1 P23141 1/20 0.46
KDM4E B2RXH2 1/20 0.45
MAPK1 P28482 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
HSP90AA1 P07900 1/20 0.44
HSP90AB1 P08238 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1581647 0.85 SLC18A3 (0.48) ALDH1A1KMT2AMAPTPOLBLMNA
SCHEMBL8596155 0.85 PARP14 (0.62) ALDH1A1PARP14PARP10HPGDKDM4E
SCHEMBL6599138 0.82 SLC18A3 (0.47) ALDH1A1KMT2AMAPTLMNAHPGD
SCHEMBL28539303 0.81 RIPK1 (0.47) ALDH1A1KMT2AHTTMAPTLMNA
SCHEMBL7729871 0.79 TSHR (0.66) ALDH1A1PARP14PARP10KMT2ALMNA
SCHEMBL24497004 0.78 ALDH1A1 (0.52) ALDH1A1KMT2AMAPTLMNAKDM4E
SCHEMBL29068350 0.78 CYP1A2 (0.57) ALDH1A1KMT2AMAPTPOLBLMNA
SCHEMBL27261597 0.77 PREP (0.55) ALDH1A1PARP14PARP10KMT2APOLB
SCHEMBL1844593 0.76 MAPT (0.55) ALDH1A1PARP14PARP10HTTMAPT
SCHEMBL16565652 0.75 SCD (0.60) PARP14PARP10HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111285872-B Indole-2-ketone derivative and preparation method and application thereof 北京志健金瑞生物医药科技有限公司 2022-05-17 CN disclosed
CN-111285872-A Indole-2-ketone derivative and preparation method and application thereof 北京志健金瑞生物医药科技有限公司 2020-06-16 CN disclosed