SCHEMBL28411784

SCHEMBL28411784

CCOC=C1C(=O)Nc2ccc([N+](=O)[O-])cc21

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 7/20 0.57
CAPN9 O14815 1/20 0.56
CASP3 P42574 1/20 0.56
CCNE1 P24864 1/20 0.56
CDK2 P24941 1/20 0.56
PDGFRB P09619 1/20 0.55
JAK3 P52333 1/20 0.55
NOX4 Q9NPH5 1/20 0.54
RET P07949 4/20 0.53
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
TGM2 P21980 1/20 0.48
EGFR P00533 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7543664 0.79 RET (0.52) PDGFRBRETMEN1KMT2ATGM2
SCHEMBL7238212 0.79 RET (0.55) RETMEN1KMT2ATGM2
SCHEMBL7238205 0.79 RET (0.55) RETMEN1KMT2ATGM2
5-Nitroisatin SCHEMBL27856567 0.75 CAPN9 (0.85) GSK3BCAPN9CASP3CCNE1CDK2
SCHEMBL11882118 0.75 SMN1; SMN2 (0.57) PDGFRBRETTGM2EGFR
SCHEMBL3752053 0.74 NOX4 (0.70) GSK3BCAPN9CASP3CCNE1CDK2
SCHEMBL1851095 0.74 RET (0.67) GSK3BCCNE1CDK2PDGFRBJAK3
SCHEMBL13080904 0.74 RET (0.67) GSK3BCCNE1CDK2PDGFRBJAK3
SCHEMBL1851097 0.74 RET (0.67) GSK3BCCNE1CDK2PDGFRBJAK3
SCHEMBL7479233 0.74 GSK3B (0.51) GSK3BCAPN9CASP3CCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111285872-B Indole-2-ketone derivative and preparation method and application thereof 北京志健金瑞生物医药科技有限公司 2022-05-17 CN disclosed
CN-111285872-A Indole-2-ketone derivative and preparation method and application thereof 北京志健金瑞生物医药科技有限公司 2020-06-16 CN disclosed